ImpiloAmalungiselelo

"Loperamide": ukubuyekezwa, imiyalelo, izinkomba ukusetshenziswa

Edinga izidakamizwa "loperamide"? Izibuyekezo ngalokhu izidakamizwa futhi izinkomba zayo, imiphumela emibi, contraindications imiyalelo izokwethulwa kulesi sihloko. Futhi, sizobe ngikuxoxele ukuthi izici kwemithi akushilo kusho ukuthi ingxenye yaso, kulokho yakha ikhishwe, njll

Ukwakheka, emabhokisini ukuma kanye nencazelo

Ngayiphi ifomu ungakwazi ukuthenga imithi efana "Loperamide"? ochwepheshe lezivakashi baphikisa ngokuthi izidakamizwa yanikezwa Pharmacy ngesimo amaphilisi, amaphilisi kanye amaconsi absorbable.

Eyokuqala amafomu amabili ahloselwe abantu abadala nezingane, eminyakeni eyisithupha eyedlule. Ngokuphathelene nalokhu kwesibili, kwamanye amazwe okuya isetshenziselwa kuphela izinsana kuze ngonyaka. Nokho, e-Russian Federation, leli fomu akuvunyelwe ukuba kusebenze, ngoba ngokuvamile isetshenziswa bebodwa, ngaphandle kadokotela we udokotela, okuvame ukuholela engathi sína, kuhlanganise nokufa.

I asebenzayo izidakamizwa zithutha futhi capsule kuphuma loperamide hydrochloride. Uphenyo odokotela sisho futhi ukuthi ingxenye kuqukethwe zombili lezi zinhlobo e esilinganayo, okusho 2 mg. Ngokuqondene izakhi eyengeziwe, zingozi zihlanganisa i-lactose, magnesium stearate, corn isitashi, talc futhi Silica colloidal.

Amaphilisi Abonayo ekhiqizwa endaweni igobolondo gelatin. okuqukethwe yabo - powder elimhlophe noma awube mhlophe. Tablets futhi abe ukuma flat futhi kungaba tint aphuzi.

Zombili lezi zinhlobo zezindlu zomuthi eziqukethwe amashashaza, okuyinto ezibekwe amakhadibhodi amabhokisi.

izici kwemithi

Liyini ikhambi njengoba "Loperamide"? Izibuyekezo kunodokotela usazise ukuthi lokhu siyefana imithi antidiarrheal.

Ngu sesibopho ukuthobisa receptor opioid izindonga emathunjini, umshanguzo izidakamizwa esebenzayo kunciphisa motility kanye ithoni imisipha abushelelezi emathunjini. Lokhu kunomthelela siyehla ukudlula elikuqukethe, futhi kunciphisa excretion of electrolyte kanye indle ketshezi.

Kufanele futhi wazi ukuthi i-ejenti kubhekwe kwandisa ithoni sphincter (anal) okwagcina ikhuthaza deceleration nesifiso sokufuna azikhulula nokugcina indle.

izidakamizwa "loperamide" Kuyoze ukusebenza ngeke? Nobufakazi bathi umphumela kokuthatha lesi imithi iza ngokushesha okukhulu. Futhi uyaqhubeka amahora 5-6.

izakhiwo pharmacokinetic

ugxile kanjani ngokushesha izidakamizwa esebenzayo kubhekwa imithi (loperamide hydrochloride)? Izibuyekezo Ochwepheshe aqukethe ulwazi emakamu elikhulu isithako esebenzayo kwaleli thuluzi kufezwa ngokusebenzisa amahora 2.6 ngemva ukungenisa. Absorption we nomuthi 40% kanye amaprotheni ngibopha - 97%.

Kufanele kuqashelwe ukuthi le izidakamizwa akusho zingene umgoqo gazi ebuchosheni. Ngaphezu kwalokho, umzimba walo cishe ngokuphelele esibindini (by lokuhlanganisa).

Inkathi isigamu-ukuphila kusho - amahora 10-14. Ithanda ke isuselwe izibilini, nezinso (ezincane okuyingxenye).

ubufakazi

Kungani ezibekiwe kusho "loperamide" izingane? ochwepheshe lezivakashi ukhulume iqiniso lokuthi lokhu izidakamizwa zingafundwa izingane nje kuphela kodwa futhi abadala. Kuhloswe for ekwelapheni lingaze sohudo ezingalapheki ne-acute zasezindaweni ezihlukahlukene (nomzimba, izidakamizwa, ngokomzwelo, kwemisebe, njll). Ngaphezu kwalokho, izidakamizwa esebenzayo uyakwazi ukulungisa kwesitulo iziguli ukuxilongwa njengoba ileostomy.

Izimo

Awukwazi ukusebenzisa imithi "loperamide" Uma kukhona izimo? Yokusetshenziswa, odokotela yangempela wazise ukuthi izimali is hhayi Kunconywa in iziguli hypersensitivity kuya izidakamizwa, ukungezwani ne-lactose, lactase ukuntula noma zikashukela-galactose malabsorption, diverticulosis, isimiso emathunjini, izilonda emathunjini esigabeni oyingozi, uhudo iphutha ngemuva enterocolitis pseudomembranous (acute).

Kufanele kuqashelwe ukuthi le imithi angeke lisetshenziswe monotherapy for uhudo nezinye izifo yaleli pheshana emathunjini, ukukhulelwa (ikakhulukazi senyanga yokuqala) kanye lactation.

Kungenzeka yini ukunikeza lesi sidakamizwa "loperamide" izingane? ochwepheshe lezivakashi bathi izidakamizwa amaphilisi izingane kungukuthi ebekiwe.

Ngokunakekela okukhulu imithi inikezwa iziguli nge esingamahlalakhona hepatic.

Izindlela kanye umthamo izidakamizwa

Indlela ukuthatha lesi sidakamizwa "loperamide" (izinkomba ukusetshenziswa, impendulo mayelana naleli thuluzi, ungathola esihlokweni samanje)?

Amaphilisi kumele kugwinywe lonke ngaphandle ukuhlafuna, ne inani elincane lamanzi. Njengoba for amaphilisi, basuke ibekwe ngaphansi kolimi. Ngemva nje kwemizuzwana, izidakamizwa kumele ziyoncibilika ngokuphelele, okwathi ngemva kwalokho proglotnut edingekayo lonke ngamathe. Tablets akufanele baphuze amanzi.

Umthamo izimali kuncike yobudala isiguli.

Ngo ukucubuluza okungapheli ne-acute zaphathwa abadala amaphilisi amabili (ekuqaleni) bese capsule 1st ngemva sezinyawo (uma kwesitulo namanje ketshezi).

Ngo-acute sohudo izingane ineminyaka engaphezu 6 ezisebusweni capsule kuqala emva ukunyakaza wamathumbu ngamunye.

esiphezulu I umthamo wansuku zonke abadala (ezingamahlalakhona kanye nesifo sohudo-acute) kuyinto 8 amaphilisi, nezingane - 3.

In the ukungabikho esihlalweni amahora angaphezu kuka-12, futhi ngemva ukuzinza, ukwelashwa ngalo muthi kufanele wayeka.

ukweqisa izidakamizwa

Yini ozoyenza kuphakama uma isiguli wathola imithi engalungile "loperamide" (amaphilisi)? Uphenyo odokotela bathi izimpawu ezilandelayo ukweqisa izidakamizwa kungenzeka kulokhu: wamathumbu isimiso, CNS ukucindezeleka (stupor amajaqamba, ukozela, kusebentisana kahle, ukucindezeleka zokuphefumula futhi imisipha hypertension).

Njengoba ekwelapheni yokwelapha lingaze. Isiguli sagezwa isisu, uyobanika isebenze namalahle.

Nge ukweqisa izidakamizwa of kweso lwezokwelapha kuyadingeka, okungenani izinsuku ezimbili.

Nokukhulelwa kanye lactation

Ngingakujabulela yini lesi sidakamizwa "loperamide" phakathi nenkathi yokukhulelwa? ochwepheshe lezivakashi wazise ukuthi ithuluzi is contraindicated ku senyanga yokuqala. Ngokuphathelene eyesibili neyesithathu, kule nkathi abesifazane imithi antidiarrheal kungenziwa ebekiwe, kodwa ngemva kokuba i ukuzimisela Inhloso isilinganiso kwemihlomulo kulabo abangamalungu akhokhela lo mama nokulimala umntwana.

Ngoba inani elincane izidakamizwa ezitholakala ubisi lwebele, kuyilapho kuzothatha ibele kufanele inqanyulwe.

side effects

Ngokuvamile, lesi sidakamizwa "loperamide 'ebekezelele ngokubhekakade kahle impela. Nokho, kwezinye izimo, isiguli bangezwa ukusabela nomzimba (isb, ukuqubuka kwesikhumba), kanye nokuqwasha noma Ngakolunye uhlangothi, ukozela, hypovolemia, isicanucanu, isiyezi, electrolyte thuthuva, gastralgia, kome ngomlomo mucosa, ubuhlungu noma kabi esiswini, ukuhlanza, emathunjini colic futhi ukubuyisa.

Kufanele kuphawulwe ukuthi kakhulu kuyaqabukela njengoba side effects e iziguli nokugcinwa urinary futhi ileus.

Izici izidakamizwa

, Kufanele uxhumane nodokotela wakho uma nomphumela oqabulayo is hhayi waphawula ngemva kwezinsuku 2 nokwelashwa izimali.

Uma ngesikhathi yokwelapha livela ukuvuvukala noma ukuqunjelwa, umuthi kufanele ayisekho. In iziguli nge kahle isibindi umsebenzi kudinga aqashelwe ngokucophelela izimpawu CNS ubuthi.

Phakathi sohudo kufanele wenze i-ukulahlekelwa electrolyte nasoketshezini.

imithi Izibuyekezo

Izibuyekezo sokulungiselela ezifana "Loperamide" lingama omuhle. Lokhu kungenxa yokuthi lokhu umuthi ngempela ngempumelelo aqede sohudo ukuthi singenzeka for yezizathu ezihlukahlukene (isibonelo, emva edilini iholide, isampula izithelo ezingavamile, ngaphambi kwaleso senzakalo ethokozisayo, njll).

Amaphilisi kanye "loperamide" capsule ayashesha kakhulu. Ngesikhathi esifanayo avumela isiguli ukuba bahlale "yokusebenza" isimo usuku lonke.

Ngaphezu ukusebenza kahle high, Inzuzo enkulu leli thuluzi izindleko zalo ongaphakeme.

Ithathwe ndawonye, zonke izinzuzo zalesi izidakamizwa waba nedumela elihle. By the way, umnikelo wakhe omkhulu kuso Unezibuyekezo omuhle labo bantu owake isicelo leli thuluzi.

Kufanele kuphawulwe ukuthi ngaphezu Plus, lokhu imithi has nezihibe. Ezinye iziguli esekhala engemihle. Nakuba, ngokuvamile, izici ngisho enjalo engemihle musa ukumosha jikelele umbono omuhle salesi sibhedlela.

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