ImpiloAmalungiselelo

"Valium" - kuyinto ... Incazelo, imfundo, isenzo nozakwabo

"Valium" - kungenxa izidakamizwa? Impendulo yalo mbuzo uzothola kancane okunye. Siphinde ukunitshela ngaloNkulunkulu ithuluzi isebenza kanjani, ukuthi izakhiwo it libhekene njengoba kufanele kube futhi kulokho yakha ikhona.

Ifomu kanye nokwakheka emaphaketheni

"Valium" - umuthi angathengwa ngesimo umjovo, kanye amaphilisi. Lokho ingxenye lezi zimali?

iqukethe 5 mg diazepam e 1 ml of isixazululo umjovo. a nomuthi okunjalo ithunyelwa 50 noma 10 amnyama ingilazi ampoules ka 2 ml, afakwe amakhadibhodi amabhokisi.

Ngokuphathelene amaphilisi, bangase aqukethe 10 noma 5 mg diazepam, kodwa futhi izithako elandelayo eyengeziwe: corn isitashi, anhydrous lactose, i-calcium stearate, isitashi pregelatinized, udayi.

Kusho "Valium" ngefomu ithebhulethi phama amakhadibhodi amabhokisi, okuyinto aqukethe Valium Valium.

Yezemithi izidakamizwa

"Valium" - umuthi ubukisa anxiolytic, miorelaksiruyuschee, sedatives, hypnotics anti-kokuquleka izakhiwo.

Ngaphambi kokuthi ngikuxoxele lo mshini wezenzo izimali, kufanele aqondwe ukuthi.

Izidakamizwa "Valium" inegama elandelayo nokuphathelene - "Diazepam". Lesi sidakamizwa kungokwalabo iqembu benzodiazepines nokuba ukubaluleka okukhulu kwezokwelapha.

"Valium" - umuthi, ngenxa yomsebenzi walo anxiolytic, aqede yangaphakathi nokukhathazeka, ukwesaba, ukukhathazeka nokucindezeleka. Ochwepheshe bathi "Diazepam" umphumela umthamo-kuncike isimiso sezinzwa esiyinhloko. Ngamanye amazwi, ngesilinganiso esincane (mayelana 2-15 mg ngelanga), lokhu izidakamizwa kubangela inkanuko umphumela, futhi ezinkulu (ngaphezu kuka-15 mg ngelanga) - ukupholisa.

Izici imithi

Kuyini ephawulekayo yindlela ngokuthi "Valium"? Action (central imisipha relaxant) zomuthi Lihlobene nokubhekana ubuso okwehlisa ikhaliphe polysynaptic emgogodleni. Ukuthola lokhu ukulungiselela kuholela ekuncipheni wegazi, ukunwetshwa izitsha yenhliziyo, kanye ngcono ukumelana hypoxia palsy futhi ngakhula ubuhlungu embundwini.

kinetics

I nomuthi "Valium" analogs okuyinto aboniswa ngezansi, amuncwa umzimba kusuka pheshana emathunjini (ngomlomo). Uma lokhu ukumuncwa kwenzeka ngesikhathi u-75% kanye emakamu esiphezulu kufinyelelwe emva 1.5 amahora.

Ukuguqulwa begazi zomuthi esibindini. Kuleli fomu le metabolite asebenzayo nge nengxenye-ukuphila. Ngo kuqokwa izidakamizwa ukuze izinsana umphumela kufinyelelwe ngemuva kwamahora angu-30, kanye nasebekhulile, kanye nabantu abadala - ngokusebenzisa 100, futhi amahora angu-48, ngokulandelana. Kulesi sibalo pathologies isibindi yesikhathi eside izinsuku 4.

ukulungiselela Okubukwe ethathwe umzimba womuntu ngokuyinhloko izinso (90%) ngesimo conjugates, kanye ingashintshiwe (2%) kanye kanye indle (8%).

ubufakazi

Ngayiphi zifo zingase isiguli kufanele inikezwa "Valium"? Izibuyekezo ochwepheshe ukubika ukuthi lokhu izidakamizwa kuboniswa ukuthola ngaphansi kwale mibandela elandelayo:

  • zibe of imisipha yohlaka ngesikhathi ukuhlukumezeka wendawo;
  • yokukhathazeka;
  • myositis, samathambo, bursitis, ukhalo-spondylitis samathambo esingelapheki polyarthritis lesichubekako;
  • ngqi;
  • umfutho wegazi ophakeme, dysphoria, isilonda esiswini kanye duodenum 12 (njengesilwane izindlela ezengeziwe), isilethikusebenza;
  • ukuqwasha;
  • angina;
  • izimo spastic, kuhlanganise i-cerebral palsy, isifo sokuqaqamba kwamalunga kanye lwamathambo imisipha ukungezwani futhi athetosis;
  • ushevu nezidakamizwa;
  • syndrome vertebral;
  • utshwala ukuhoxiswa syndrome ne ezinjalo nokukhathazeka, ukungakhululeki, ukuyaluza, eliqhaqhazelayo;
  • isimo epilepticus, ekwelapheni ukuquleka;
  • iziyaluyalu zengqondo e zabesifazane kanye zokubelethisa (isib, menopausal futhi kokuya esikhathini, gestosis, ukuba lula zabasebenzi);
  • eczema nezinye izifo ukuthi ahambisana ukulunywa kanye nobuhlungu;
  • nesifo i-Meniere sika ;
  • isimo hallucinatory-Paranoid, motor excitation zasezindaweni ezihlukahlukene (e wezifo zengqondo kanye Neurology);
  • ukubulawa kwezinzwa okuvamile futhi premedication (isib, ngaphambi nje kokuba ahlinzwe futhi izinqubo endoscopic).

Izimo

Uma akufanele usebenzise lesi izidakamizwa ngokuthi "Valium"? Umthelela kulo muthi akufani njengoba singathanda, uma wamukela ke:

  • e hypersensitivity;
  • ikhoma, ukushaqeka;
  • acute utshwala ukudakwa;
  • amafomu acute izifo kwesibindi;
  • myasthenia gravis;
  • engela-Ukuvalwa ukufiphala;
  • kubantfwana labancane kunalabo izinyanga 6;
  • ngesikhathi lactation, futhi senyanga yokuqala sokukhulelwa.

Umuthi 'Valium ": yokusetshenziswa

Yetha kubhekwa indlela kumele kube uchwepheshe abanolwazi. Ezigulini omdala umthamo zomuthi ngemva kokuphathwa ngomlomo kufanele kube 5-20 mg ngosuku. Lokhu ngobungako izidakamizwa kunqunywa kuye kobukhulu izimpawu isifo, kanye isithombe Imininingwane emtholampilo.

Umkhawulo kungenzeka ukuphathwa umthamo akuyona engaphezu kuka-10 mg. ukwelashwa Yiqiniso lokhu kusho esimweni yokukhathazeka kufanele liqhubeke 6 amasonto. Emva kwalesi sikhathi kufanele ubheke udokotela ukuya, kangangokuthi kwadingeka izinhloli imali yesondlo umthamo ubuncane.

Ukuqedwa umuthi kancane kancane kubhekwa.

Ezimweni eziphuthumayo, nomuthi asebenzayo ukuba parenterally (intramuscularly noma ngemithambo yegazi) iqondiswa. Kulokhu, umthamo we 2-20 mg.

Nge ukumnika emthanjeni zomuthi kufanele sinikezwe kancane, ngesilinganiso esingeqile 0.5-1 ml ngomzuzu.

side effects

Njenganoma iyiphi imithi, ukuthatha olucutshungulwayo izidakamizwa kungabangela ukusabela. Lezi zihlanganisa lokhu okulandelayo:

  • bradycardia noma hypotension;
  • kwehle okuhlushwa izinga yokusabela;
  • ukuluthwa izidakamizwa;
  • isiyezi kanye ikhanda;
  • ukuthuthukiswa ukusabela nakuba yokukhathazeka, ukuqwasha, ukusangana, kanye nokuquleka;
  • inkumbulo ukungakhuli (dlala);
  • ukusabela ohlangothini kusayithi umjovo;
  • ukunyakaza iziyaluyalu ezifana dysarthria futhi ataxia;
  • ukulimala nezinso isibindi, esiswini atony, kwehle libido futhi potency (ukusetshenziswa eside zomuthi);
  • komzimba;
  • ukuhoxiswa syndrome;
  • kwehle ukusebenza, futhi ukuba buthakathaka kwezicubu.

Ngo ukuqokwa izidakamizwa isiguli kubaluleke kakhulu ukwazisa kwakhe ukuthi lena izidakamizwa. Ngemva kubhekwe owaziwayo psychotropic ejenti imijovo, okuyinto has eziningi nemiphumela engemihle, phakathi okuyinto ikakhulukazi walulama umlutha kanye zokuqaleka.

UDkt zimise lo muthi ubophekile ukuba wazise nesineke ngemiphumela ebuhlungu izidakamizwa emzimbeni wakhe, kanye sipho nezinye izindlela zokwelapha.

ukweqisa izidakamizwa wezokwelapha

Overdosing kubhekwe izindlela ezingemnandi ephelezelwa izimpawu ezifana CNS ukucindezeleka. Isenzakalo esifanayo angase abe kobukhulu obuhlukahlukene, ezisukela ukozela nesiphetho equlekile. Futhi, uma nithatha ebulilini izidakamizwa hypotension lesiguli kungenzeka, ukudideka kanye nokucindezeleka zokuphefumula.

Ukwelashwa izimo ezinjalo nge ngalo mbandela, uma isiguli sifuna bayazi, kuhilela lokungeniswa ka emesis kanye nokusetshenziswa kwe-carbon isebenze. Kuleso simo, uma isiguli aquleke, ke sagezwa esebenzisa uphenyo esiswini, kanye yokwelapha lingaze, ukuhlolwa imisebenzi ebalulekile kanye nokwethulwa uketshezi ukuthuthukisa diuresis.

Ukuze asebenze ngokuzimisela ukuze kuboshwe ukuyaluza ngokweqile isiguli, unganikezela ke barbiturates.

Ukuxhumana nezinye izindlela zokwelapha

I nomuthi "Valium" kubangela potentiation utshwala imiphumela, hypnotics, anticonvulsants, ama-ejenti hypotensive futhi antihistamine, futhi antipsychotics, imithi ebulala izinzwa jikelele, tricyclic antidepressant, imisipha relaxants futhi analgesics.

evuselela Analeptic futhi kungaba kakhulu ukunciphisa umsebenzi "Diazepam" izidakamizwa.

Antacids wehlise izinga, kodwa hhayi ezingeni ukumuncwa zomuthi.

inhibitor okunjalo ka microsomal namachibi ngokuthi "Cimetidine", "Omeprazole" "ketoconazole" "fluoxetine" futhi "Fluvoxamine" siguqula pharmacokinetics zomuthi akhuluma ngayo, futhi ukwandisa isikhathi yemiphumela yayo emtholampilo.

"Rifampicin" kunciphisa lokuhlushwa "Diazepam" egazini, "Erythromycin" kubambezela umzimba walo esibindini.

izidakamizwa ezifanayo

Yini engathatha isikhundla sale izidakamizwa ngokuthi "Valium"? Analogue eRussia kungukuthi edayiswa Pharmacy. Ngaphezu kwalokho, le mithi kokudedelwa kuphela ngemva kokwethula kadokotela.

Buyisela izidakamizwa can "sibazon", "diazepam" noma "Diapamom". Nokho, lokhu kufanele kwenziwe kuphela emva kokubonisana udokotela.

Lokho okwakudingeka ukuze kukhokhwe izidakamizwa

Njengoba ngishilo ngenhla, ukuthenga izidakamizwa "Valium Roche" eRussia Ngeke zonke ekhemisi. Izindleko zomuthi - ruble abangaba yinkulungwane (iphakethe ngalinye).

Intengo imali e-UK nakwamanye amazwe aseYurophu, ngokuvamile mayelana amabili namashumi amahlanu esingamakhilogremu ngamunye amaphilisi ayizinkulungwane (10 mg).

Ukuze uthenge emzini buyisidakamizwa enjalo ukuthi uzohlangana zonke izidingo zokuphepha kanye nekhwalithi, ochwepheshe batusa ukuba zisebenze ngemuva, lapho uzonikezwa ulwazi olugcwele ukutholakala kwayo Pharmacy kanye namanani nenzuzo kakhulu mayelana.

Umthengi izibuyekezo mayelana nemithi

"Valium" - kuba zithandwa iziguli umuthi isetshenziswa njengenhlangano anxiolytic, miorelaksiruyuschego, sedatives, hypnotics, futhi anticonvulsants. Ngokusho ngempendulo iningi abathengi, kubhekwa umuthi kakhulu izifo ezihlukahlukene, kuhlanganise nesifo sokuwa, izinkinga zokulala, ukukhathazeka nokunye. Futhi ukuthatha kuyasiza ekudambiseni izimpawu njengoba ukuyaluza, eliqhaqhazelayo nekugwema ngamaphupho nje la.

Nokho, akukho ithuluzi ezifana owawuzovumelana wonke umuntu. Abanye abantu abasebenzisa lesi izidakamizwa abangajabule. Bona wazi ukuthi izidakamizwa iqala ukwenza kuphela ngemva kwesonto. Ngaphezu kwalokho, nge ukusetshenziswa okuqhubekayo the nomuthi kubangela inani elikhulu ohlangothini ukusabela kanye kuholela ekubeni umlutha wezithombe.

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