ImpiloAmalungiselelo

Imiyalelo Isicelo, impendulo Analogue "Locri"

Abanomfutho wegazi ophakeme nesifo senhliziyo kuvamile emhlabeni. Lesi isifo sasivumela kunganakekile, okuyinto kusaqalwa kunzima ukukhomba. Ngakho ngemva kweminyaka engu-40, kufanele ukuqapha njalo dvleniya ukusebenza. Uma imiphumela ephezulu kakhulu, kufanele uxhumane nodokotela wakho. I ngaphambili ukwelashwa siqala, ngokushesha onganqoba sifo.

izidakamizwa Modern zinezikhathi ukusebenza kahle eliphezulu. Leli qembu ukuvimba. Tablets ngobumnene kakhulu kunciphise umfutho wegazi futhi akulimazi umzimba. Ethandwa kakhulu phakathi abelaphi namuhla belungiselela "Lokren". Yokusetshenziswa, analogs, umthamo efanele - konke lokhu kwaziswa lapha ngenzansi.

Ukwakheka kanye nefomu wokukhulula izidakamizwa

Tablets "Lokren" amhlophe, kancane ayizindunduma ngakolunye uhlangothi ephawulwe okudweba nombhalo othi EK20. With titer ezinjalo zemithi kungaba avelele kalula kusuka mbumbulu. Izibhebhe embozwe igobolondo mncane. Isakhi esiyinhloko lichaza ekwakheni izibhebhe kubhekwa gidrohrorid betaxolol mg 20. Nezinsizasenzo mithi monohydrate lactose, cellulose ezincane, i-sodium karboksilmetilkrahmal.

Igobolondo yakhiwa gipromilozu, macrogol, ama-titanium dioxide. Itholakala amaphilisi ngendlela ibhamuza, futhi izingcezu 14 ngamunye. Noma yimuphi Analogue "Locri" uyoba ukwakhiwa efanayo futhi izinkomba ukusetshenziswa.

Imiphumela izidakamizwa emzimbeni

Tablets basonta iqembu beta-blocker. Basuke libhekwe njengelingcwele blocker abakhethayo lomugqa wokuqala. Betaxolol, okuyinto ingxenye izidakamizwa, has cardioselective beta-adrenoceptor Ukuvinjwa umphumela, libhekene zingenzi lutho olunyakazisa agonist kuyinto ulwelwesi ababuthakathaka. Ngenxa yalesi izidakamizwa encishisiwe kwenhliziyo ngesikhathi umsebenzi ukuphumula kanye ngokomzimba. Umthelela main - kunciphisa umfutho wegazi uphumule futhi lapho uvivinya umzimba.

Uma usebenzisa izidakamizwa sihamba tachycardia, encishisiwe umthwalo inhliziyo, evamile neuropathy kwegazi. inciphise umfutho wegazi ophakeme ka betaxolol ngokusebezisa isikhathi eside akuyona encishisiwe. Lapho ezibhebheni ukungenisa umthamo owodwa umphumela zokwelapha kwenzeka phakathi namahora amathathu futhi uyaqhubeka usuku lonke. Imiphumela Esitebeleni ingatholakala nge Yiqiniso Clusive yokwelashwa. Izenzo ezinjalo sigqoke amaphilisi umzimba "Lokren". Izidakamizwa analogue futhi normalizes izinkomba igazi lapho kusetjentiswe kahle.

Pharmacokinetics

Lapho udle, umuthi ancibilikisa ngokushesha futhi ngo-100% ugxile kusukela esiswini. Umthelela esiphezulu kufinyelelwa ngemuva kwamahora amabili e-plasma. Umuthi sibopha ukuthi igazi eligciniwe ngo-50%. Betaxolol e isibindi lwakha metabolites esingasebenzi. Cishe u-80% isithako esebenzayo excreted ngu izinso ngesimo metabolites. 20% livela umzimba zinjalo.

Fast ngokwanele kungenzeka kuzuzwe nomphumela zokwelapha omuhle, uma ukuthatha kahle amaphilisi "Lokren". Yokusetshenziswa aqukethe lonke ulwazi oludingekayo.

Izinkomba kanye contraindications

Isizathu ukuqokwa zomuthi kubhekwa nomfutho wegazi ophezulu. Kusho zingafundwa eyedwa noma inhlanganisela neminye imithi ukwehlisa ingcindezi. Tablets babelwa ukuze kuvinjelwe imivimbo ngesikhathi.

Izimo emithini yokuselapha kubhekwa ezinzima somoya bronchial kanye ukucinana kwemithambo yomoya emaphashini, ukwehluleka oyingozi inhliziyo. Musa ukuphuza imithi ngesikhathi uzwakalise imihlola bradycardia, amafomu okunzima isifo Raynaud sika kanye neuropathy ukuphazamiseka kwegazi. Kukhona imikhawulo yobudala. Imithi engamiswanga iziguli ezincane.

It is hhayi Kunconywa ukuba baphuze amaphilisi in iziguli esingamahlalakhona kwezinso noma hepatic. Ngesikhathi ekhulelwe futhi ithuluzi lactation ingasetshenziswa kuphela uma inzuzo ezingase zisetshenziselwe ukuba umama idlula ingozi ezingase zisetshenziselwe ukuba usana.

Ngaphambi ukwelashwa kufanele ufunde ngokucophelela imiyalelo ukusetshenziswa kwezimali "Lokren". ochwepheshe lezivakashi basikisela ukuthi imiphumela emibi kaningi kwenzeka kulezo ziguli musa zithobele izincomo.

Isikali

Umuthi kumele zithathwe nge nangokuphuza uketshezi oluningi. Umuthi akufanele ezokuhlafunwa. Ukwelashwa kumelwe siqale ithebhulethi isigamu (10 mg). Uma nomphumela oqabulayo omuhle, kubalulekile ukwandisa umthamo akezi amasonto amabili. Izinga sangemihla ayikwazi ukudlula 40 mg.

Odokotela abaningi musa batusa ukuba iziguli zabo baphuze iphilisi ezingaphezu kwesisodwa ngosuku. Uma une abampofu ingcindezi kwehliswa afanele ukwengeza elinye ukwelashwa izidakamizwa antihypertensive. Iziguli ezinzima esingamahlalakhona kwezinso kufanele uqale ukuthatha izidakamizwa umthamo 5 mg. Kancane kancane ukwandisa izinga nsuku zonke. It has ukuba zihlolwe ngaphambi kokusebenzisa izindlela "Lokren" imfundo manual.

ukweqisa izidakamizwa

Nge ukweqisa izidakamizwa amaphilisi bangezwa inzululwane, ophezulu iconsi, cyanosis yeminwe nezinzipho, bradycardia, lightheadedness. Futhi nezimpawu ezifana bronchospasm futhi senhliziyo.

Ukwelashwa nokuvikelwa kokudla siqukethe lavage esiswini. Kunconywa ukuthi uphuze adsorbent nesineke futhi axhunyiwe yokwelapha ukumnika. Ngo ukwehla olukhulu endleleni ingcindezi kuyadingeka ukuze prokapat "Dopamine" bese ufaka "Atropine". Kufanele nakanjani wengeze glycosides inhliziyo futhi antispasmodics. Ezimweni ezimbi kakhulu, ekubonisa ukwethulwa igazi esikhundleni ne-plasma. Noma yimuphi Analogue "Locri" Kufanele uthathe, kulandela umthamo ebekwe udokotela.

side effects

Lapho nokwelapha izidakamizwa yokusabela iguliswa zingaqala. It kubonakala ngesimo ukuqubuka esikhumbeni futhi ukulunywa. Futhi, kukhona ukusabela phezu ingxenye isimiso sezinzwa, okuyinto kuboniswa isiyezi, ubuhlungu bekhanda, asthenia, ukuqwasha, amaphupho amabi, paresthesia. Imiphumela engemihle zibandakanya kwehle umbono, bese wehlise ingcindezi intracranial. Ngesikhathi ukuthatha amaphilisi sivame ukuba ubuhlungu besisu, isicanucanu, ukuhlanza. Kwangathi shintsha igazi nokuthuthukisa leukopenia. Abesilisa ngokuthatha izidakamizwa kubangela nokuvusa induku. I ngokuqapha kufanele aqokwe amaphilisi kakhulu eminyakeni yokuguga.

Kumele ligcinwe ngaso ekamelweni lokushisa endaweni emnyama ezingafinyeleleki izingane, lesi sidakamizwa "Lokren". Analogs elisetshenziswa izimo ezifanayo.

Analogue "Locri" eRussia - isidakamizwa "Betaxolol"

Indlela ukukhetha esikhundleni izinga imithi? Kuthiwani uma ekhemisi ayengenayo indlela "Lokren"? Izidakamizwa analogue uzokwazi ukuncoma udokotela njalo. izindlela ezidumile "Betaxolol." It cardioselective beta-blocker esetshenziswa kunciphise umfutho wegazi nokuhlasela angina. Ngemva kokungenisa wajinge wanamatsela esiswini ngokuphelele. Umthelela esiphezulu kufinyelelwa ku-plasma amahora amathathu. Umuthi excreted ngu izinso ngesimo metabolites ukuthi akhiwa esibindini.

Umuthi kwehlisa ingcindezi intraocular kahle, uma usebenzisa ikhambi ngesimo iso amaconsi.

Umuthi isetshenziswa kanye ngosuku ngesikhathi umthamo mg 20. Imithi zingafundwa wedwa noma njengengxenye ukwelashwa. Akunconyelwe ukusetshenziswa phakathi nokukhulelwa kanye lactation. Ezimweni ezingavamile, izidakamizwa kubangela imiphumela eminingi engemihle njengezindlela ngesimo ukuqubuka kanye ukuncinza esikhumbeni. Futhi, kungase kube isiyezi kanye nesicanucanu, kanye besebenzisa amaphilisi "Lokren". Russian analogue abe izinkomba efanayo kanye contraindications.

Izidakamizwa "Betacam"

Imithi kungokwalabo beta-blocker emgqeni wokuqala. amaphilisi emhlophe. umthamo ngamunye equkethwe mg betaxolol hydrochloride 20. Imithi kungenziwa kunqunyiwe ngudokotela. Lesi sidakamizwa sisiza kulesetayelekile blood pressure, ukunciphisa kwenhliziyo uphumule futhi ngesikhathi umsebenzi, kuholela evamile neuropathy kwegazi futhi aqede angina.

Akunconyelwe imithi e pathologies we nezinso isibindi. Phakathi nokukhulelwa kanye lactation izidakamizwa akuvunyelwe. Agent bangase baxabane nomzimba futhi ngeziphambeko omncane izinhlelo sezinzwa futhi wokugaya ukudla. Okumele kuqashelwe kufanele libekwe abantu lapho usukhulile futhi uma hypersensitivity kuya izingxenye ezibhebheni. Lokhu Analogue "Locri" Ungashintshanisa ngokuphelele amazwe yasekuqaleni.

Izibuyekezo

Mayelana Beta-blocker ochwepheshe sokukhuluma kahle. Isikhathi esifushane kungenzeka kulesetayelekile kwemigomo ingcindezi nokwehlisa kwesokunxele ventricular hypertrophy. Le mithi bubekezelelwa kahle futhi akuphazamisi umsebenzi nezinye izitho neenkambiso. Noma yimuphi Analogue "Locri" kuzobonisa nomphumela omuhle uma isetshenziswa ngokuhambisana nemiyalelo.

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