ImpiloAmalungiselelo

Tablets "Agalates": ukubuyekezwa, yokusetshenziswa, intengo

Kanjani lesi sidakamizwa "Agalates"? Izibuyekezo ngalokhu izidakamizwa, sizobe ukwethula e mathiriyeli lo sihloko. Uyofunda indlela yokusebenzisa nomuthi wathi, ukuthi kubiza malini, uma unanoma yimiphi imiphumela emibi kanye contraindications, okuyiwona wona kuhloswe, nokunye.

Ukwakheka, emabhokisini akha wedivaysi yezokwelapha

Ngayiphi ifomu senziwa imithi "Agalates"? ochwepheshe lezivakashi bathi umuthi onjalo kungatholakala Pharmacy kuphela ifomu tablet. nempahla yabo esebenzayo cabergoline. Futhi, izidakamizwa kuhlanganisa i-lactose, L-leucine kanye magnesium stearate.

Thenga amaphilisi "Agalates" (intengo, ukubuyekezwa abekwe ngezansi) kungaba in dark ingilazi izimbiza, okuyinto ezibekwe inqwaba amakhadibhodi.

kwebalingisi kwemithi zomuthi

Tablets "izilinganiso Agalates 'zazo axutshwa, kukhona zokwenziwa ergot alkaloid. I-ejenti asebenzayo zomuthi liziphatha njengenhlangano agonist ka Dopamine receptor. It kuvimbela prolactin uketshezi inkanuko hypothalamic dopaminergic receptor.

Isenzo zomuthi olucutshungulwayo kuncike umthamo. Ukwehla prolactin egazini kwaba mayelana 3 amahora futhi kuthathe amasonto 2-3.

Phakathi ekwelapheni hyperprolactinemia ezingabantu kanye bubuhle ubulili prolactin okuqukethwe ngokuvamile kwesejwayelekile emva 3-4 amasonto.

izidakamizwa "Agalates" Indlela Isebenza? Imiyalelo, amazwana kusukela ochwepheshe usazisile ukuthi leli thuluzi kunomphumela abakhethayo kakhulu. Kulokhu, kuba ngokuphelele ephephile futhi kuqhathaniswa asibekezeleleki kahle.

Asinakusho ukuthi ngenxa kokuthola kuhlolwe amaphilisi iziguli zingase zibhekane ukwehla komfutho wegazi. Ngaphezu kwalokho, izinga kwawo kuxhomeke kulokho umthamo. Prakthiza ebonisa ukuthi umphumela hypotensive laligujwa amahora kuphela ngemva kuka 6 (ngemva reception).

Izimfanelo pharmacokinetic zomuthi

Manje uyazi ukuthi kuyinto izidakamizwa "Agalates". Imiyalelo, intengo, ukubuyekezwa mayelana izidakamizwa ekulesi sihloko.

Ngemva kokuphathwa ngomlomo, izidakamizwa ngokushesha ngempela ugxile kusukela pheshana emathunjini. Ngo igazi lomuntu kunqunywa ngemuva kwamahora mayelana 1-4. Mayelana 42% yemali nakanjani plasma amaprotheni.

Cishe zonke metabolites cabergoline uqale zivimbela ukukhiqizwa prolactin, kodwa kuphela ngezinga elincane. Impilo kwesigamu umuthi cishe amahora angu-80 (amahora 114 in iziguli hyperprolactinemia).

Esikhathini umchamo isiguli ukuba wayekhuluma nobani ezinqunyiwe izidakamizwa, le nomuthi itholakala isamba 18% umthamo olusetshenzisiwe, endleni - mayelana 72%.

Izinkomba ukusetshenziswa zomuthi

Yini ukuthatha amaphilisi "Agalates"? Izibuyekezo ongoti abanolwazi sincome izinkomba ezilandelayo:

  • hyperprolactinemia;
  • amenorrhea, anovulation, galactorrhea futhi oligomenorrhea, okuyinto zihlobene ngokuqondile hyperprolactinemia;
  • hyperprolactinemia idiopathic;
  • prolactin-secreting ingozi pituitary adenoma ;
  • oligomenorrhea, elingacacisiwe.

Kufanele kuqashelwe ukuthi le imithi ezinqunyiwe ukucindezela kwangemva kokubeletha lactation noma usumisiwe.

Izimo ukusetshenziswa imithi

Hlobo luni Izimo kufanele bazazi isiguli ngaphambi kokusebenzisa umuthi "Agalates"? Uphenyo odokotela ikakhulu ukhombe imikhawulo elandelayo:

  • hypersensitivity kuya izingxenye zomuthi;
  • nomfutho wegazi ophezulu kwangemva kokubeletha;
  • zokungezwani ne-lactose;
  • iziyaluyalu kwesibindi;
  • sengqondo emlandweni;
  • usakhula (iminyaka engu-16);
  • eclampsia futhi pre-eclampsia;
  • isicelo amanxusa ama-antibiotic - macrolides;
  • izilonda valvular elafika ngokumelene okwenza yokwelapha cabergoline.

Izidakamizwa "Agalates": yokusetshenziswa

Inani, izibuyekezo ngalokhu nomuthi ungabona khona kanye ekupheleni sihloko. Ngokuphathelene kulesi sigaba, khona-ke siyobe ngikuxoxele kanjani ukusebenzisa izidakamizwa ngaphansi ukucatshangelwa.

Ukuze ekwelapheni hyperprolactinemia iqondiswa 0.5 mg ngeliviki. Take it ngezinyathelo elilodwa noma amabili. Ngemva kwalokho, umthamo ukwandisa. Phakathi nenyanga yokuqala ukwelashwa kungase inani nomuthi lenyuke ngomunye 0.5 mg.

Uma usebenzisa ezingaphezu kuka-1 mg izidakamizwa ngeliviki, kumele ihlukaniswe izikhathi eziningana (2-3). Omkhulu Kunabo umthamo masonto onke kuba 4.5 mg. Njengoba ukwesekwa esetshenziswa 1 mg.

Kufanele kugcizelelwe ukuthi isipiliyoni kokuphatha lokhu kusho asebekhulile (engaphezu kwengu-65) engakaze wafunda. Ngakho-ke, ingabe kufanele ngithathe imithi kulonyaka, kungenzeka kuphela ngaphansi kweso lwezokwelapha esiqinile.

Ngenxa nomuthi "Agalates" kufanele sisetshenziselwe nezinye izinkomba? Izibuyekezo (lactation ekunqanyulweni kwenzeka ngemva kokwamukela izibhebhe 1st) ochwepheshe bathi uthatha ithuluzi ezifana kuyadingeka kuphela emva kokubonisana onguchwepheshe (obelethisayo). Ukumisa esungulwe ngokuphelele lactation nomuthi iqondiswa ngezilinganiso ka 0.25 mg kabili ngelanga. Thatha le imithi kufanele kube izinsuku ezimbili.

Uma ufuna ukuyeka lactation emva kokubeletha, isiguli kunikezwa 1 mg zomuthi ngokushesha emva kokuzalwa.

Izimpawu ngokweqile zomuthi "Agalates"

Kuze kube manje, akukho amacala overdosage aye alotshwa. Nakuba esimweni semali umuthi ematfuba emesis, isicanucanu, sengqondo, ukuhhema noma ukwehlisa wegazi. Lapho waveza uphawu overdosing kudinga ukunikezwa imithi efana "Domperidone" futhi "bromopride".

imiphumela emibi ngemva kokwamukela nomuthi

Yiziphi imiphumela emibi zenzeka ngemuva nokuphathwa kwezimali? Uma izidakamizwa isetshenziselwa ukucindezela noma ukuvimbela lactation, iziguli engaveza imiphumela enjalo enqabayo eyavezwa isiyezi, isicanucanu, ubuhlungu bekhanda, ubuhlungu besisu, ukwehla okuncane blood pressure kanye ukozela.

Ngezinye iphilisi njalo (ekwelapheni hyperprolactinemia) Kungase kudingeke ubuhlungu bekhanda, ukukhathala, isicanucanu, isiyezi, kolwelwesi, dyspepsia, ukuqunjelwa, ubuhlungu besisu, webele ngesisa, ukuhlanza, umfutho ophansi wegazi, "tide", ukucindezeleka futhi paresthesia.

Uma impatho "Agalates" izidakamizwa imisiwe, sinombono amaphilisi eside reception iziguli zingase esekhala okulandelayo side effects:

  • ukuqubuka kwesikhumba;
  • izinkinga zokulala, ukusangana, ukuba nesiyezi, ubuhlungu bekhanda, ukozela, kukhuphuke libido, ukucindezeleka;
  • isicanucanu, dyspepsia, ubuhlungu besisu, ubuhlungu esifundeni epigastric, ukuqunjelwa, ukuhlanza;
  • iziyaluyalu kwesibindi;
  • palpitations, hypotension, pericarditis nge effusion, angina, valvular isifo senhliziyo, edema neuropathy;
  • ukukhathala, asthenia;
  • effusion pleural, dyspnoea;
  • umbono kahle.

izidakamizwa ekuhlanganyeleni

Tablets "Agalates 'akufanele bathathe ngokuhlanganyela abamelene ka Dopamine receptor ezifana" Phenothiazine "," Metoclopramide "futhi" thioxanthene ".

Kufanele kuqashelwe ukuthi akuvunyelwe ukuba linqume izidakamizwa ne macrolides. Lokhu kungenxa yokuthi kukhona amathuba olukhulu anda cabergoline lokuhlushwa igazi. Ngaphezu kwalokho, it is hhayi Kunconywa ukuthatha izidakamizwa isikhathi eside kanye nezinye alkaloids ergot.

Nge ekhethekile ngokuqapha "Agalates" ithebhulethi iqondiswa kanye antihypertensives. Izidakamizwa ekuxhumaneni ne "levodopa" ayitholakalanga.

izincomo ezithile

Ngokuqapha izidakamizwa "Agalates" ekhethekile ebekwe iziguli Raynaud Syndrome, isifo senhliziyo, isilonda peptic ka ipheshana wokugaya ukudla, ukuphazamiseka we nezinso, ukopha zangaphakathi, iziyaluyalu kakhulu engqondweni emlandweni, kanye reception antihypertensives.

Ukuze kuvikelwe noma ukucindezelwa of lactation is hhayi Kunconywa ukuba linqume izidakamizwa iziguli preeclampsia futhi ngesikhathi nomfutho wegazi ophezulu kwangemva kokubeletha.

Izidakamizwa "Agalates": Izibuyekezo

Ukunqanyulwa lactation (kudingeka sithuthele ngaphambi kokuthatha amaphilisi) yilona olubonisa ezinkulu ukusetshenziswa kwalesi izidakamizwa. Ngokusho izimpendulo iziguli, lokhu izidakamizwa siyasebenza ngempela ukuba sibhekane ngokuphumelelayo nanoma yini lo msebenzi.

abesifazane abaningi abane-hyperprolactinemia ukukhuluma ka nomuthi "Agalates" kuphela ohlangothini oluhle. Ngokusho kwabo, imithi oyinikiwe nale izidakamizwa kuholela oda cishe zonke cwaningo.

iziguli futhi ukuthi le izidakamizwa ludluliselwa kubo kuhle. Nokho, zikhona izibuyekezo, lapho ucansi bubuhle esekhala isiyezi kanye nekhanda. Kulokhu, odokotela batusa imithi noma ukhansele noma esikhundleni salo iphephe kuwo izindlela zempilo.

Kungakanani buyisidakamizwa "Agalates"? Lokhu umuthi ngempela eqolo. Pharmacy eMoscow nesifunda eMoscow intengo izibhebhe ezimbili 0.5 mg zingahluka kusuka ruble 330 kuya 470.

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