ImpiloAmalungiselelo

"Elefloks": yokusetshenziswa, nozakwabo yangempela

"Elefloks" kuyinto iqembu fluoroquinolone. Ukulungiswa kuyalithinta imithi elwa nawo. The main izidakamizwa ingxenye - levofloxacin. Isixazululo kanye amaphilisi "Elefloks" kuboniswe tesikhumba, izinqubo ezithathelwanayo ngo kwezicubu ezithambile, septicemia, inyumoniya, prostatitis omsakazo webhaktheriya, sinusitis acute kwezinye izifo kanye nemvelo ezithathelwanayo.

Ukwakheka kanye uhlobo "Elefloksa" izidakamizwa

Umuthi itholakala amafomu amabili Isikali - Tablets (ukupakisha 5 no-10 nama-PC.), Isixazululo intravenous (100 ml flasks). Isixazululo equkethe 5 mg / ml isithako esebenzayo. Izibhebhe ungase wakhiwe abantu 250 noma 500 mg ingxenye eyinhloko.

Ukwakheka izibhebhe zihlanganisa ezinye excipients: polysorbate 80, magnesium stearate, crospovidone, hypromellose, MCC (Avicel-PH 101, 102).

Ama-antibiotic "Elefloks" ngesimo amaphilisi camera amaphilisi, okuyinto asetshenziselwa ukwakha yensimbi oxide (ophuzi, obomvu), macrogol, ama-titanium dioxide. Isixazululo njengenhlangano ingxenye asizayo iqukethe sodium hydroxide, amanzi umjovo, hydrochloric acid dextrose anhydrous.

isinyathelo kwemithi "Elefloks" izidakamizwa

isithako ezicindezelayo nomthelela synthesis DNA virus. izinguquko morphological kuyothi kuthinte cytoplasm, ulwelwesi kanye cell udonga nezilwanyana ezincane okubangela ukufa kwabo. Lezi zinqubo unikeze amagciwane nemiphumela imithi elwa nawo. Kwamanye izidakamizwa anaerobic singangena futhi aerobic (igremu-HIV, amalutshwana-negative), namanye amagciwane.

Iyasebenza temlomo izidakamizwa "Elefloks" ingxenye thuluzi ngokushesha ugxile kusukela ipheshana emathunjini cishe ngokuphelele. Ngezinye izilinganiso 500 mg isithako bioavailability cishe ngamaphesenti angu-100, ne-plasma yokubopha - ngesilinganiso samaphesenti angu-35 ka-. Umuthi lingena kahle kwezinye izicubu kanye izitho. Encane okuyingxenye is oxidized deacetylated yi isibindi. Ikakhulu ukuqedwa izidakamizwa kusukela umzimba eziphathelene nezinso.

Izinkomba "Elefloks" ukulungiselela

"Elefloks" analogue asetshenziswa Izilonda, prostatitis, isifo kuthinta ipheshana zokuphefumula, izitho ezakha uhlelo urinary. I nomuthi isetshenziswa njengenhlangano yokwelapha adjunct ngesifo sofuba, ogama ukuma kuchazwa njengoba esitebeleni.

Izidakamizwa ukwelapha izifo ezithathelwanayo kanye ukuvuvukala okubangelwa umthelela ongemuhle nezilwanyana ezincane ezingafani luvelo levofloxacin. "Elefloks" imfundo on isicelo ikuvumela ukwabela lapho libanjwa:

  • prostatitis kuyinto omsakazo webhaktheriya;
  • sinusitis ngefomu acute;
  • izifo naphakathi-besisu;
  • ukucinana kwemithambo yomoya emaphashini iloliwe ukuma;
  • izinqubo ezithathelwanayo ngo ngomgudu womchamo noma ngaphandle yezinkinga;
  • ukutheleleka ezithinta isikhumba nezicubu ezithambile;
  • umphakathi-atholwe i-pneumonia,
  • isifo esithinta eliphezulu izitho zokuphefumula;
  • septicemia;
  • bacteremia;
  • sofuba amelana isenzo izidakamizwa (isiqu esithi "Elefloksa" wenziwa ngokusebenzisa ukwelashwa eziyinkimbinkimbi).

Izimo ethola "Elefloks" izidakamizwa

Ukuze izidakamizwa kukhona eziningi Izimo. "Elefloks" yokusetshenziswa ayikuvumeli ukusetshenziswa e yisithuthwane ngokulandelana kwawo, iziyaluyalu convulsive, ingane esindayo kanye lactation. Umuthi lifakwa esigulini, ogama yobudala engaphansi kuka-18 ubudala. Izimo zihlanganisa umsipha ukulimala, okuyinto eyaba okushiwo quinolones yokwelapha, anda kuvelana izingxenye izindlela. Ngakho-ke, ngaphambi kokufaka isicelo kumele uzifunde ngokucophelela izidakamizwa futhi uthintane onguchwepheshe.

Ngesikhathi sokwelashwa kudinga ukubhekelwa ngokuthi isiguli ukuphulwa emsebenzini izinso, ukuntula glucose-6-phosphate dehydrogenase. Phakathi ekwelapheni iziguli esezikhulile futhi kudingeka kweso lwezokwelapha.

Ukusetshenziswa "Elefloks" izidakamizwa

"Elefloks" analogue Kunconywa ukuba asebenzise phakathi ukudla noma phambi kwabo (imizuzu engu-30 ngaphambi kokuba ukudla). Izibhebhe zingafundwa kuphela njengoba lonke ifomu isamba elanele amanzi afudumele.

Empeleni, lapho besanda kuqala ukwelashwa zonke izidakamizwa usuku ngekucikelela kuhambisana Isikhawu 1-2 amahora. Umthamo kuncike isifo, kobukhulu nenkambo ukuzwela yayo ngokwemvelo kulesi sifo izidakamizwa lwegciwane.

Ngokuvamile, lapho creatinine imvume enkulu kuka-50 ml / imiz, izinhlobo zemithi ezifana isicelo:

  • yezinkinga ukucinana kwemithambo yomoya emaphashini - umthamo ngosuku - 250-500 mg, a esiqhubeka isikhathi esisuka esontweni elilodwa kuya ezinsukwini eziyishumi;
  • egeleza sinusitis acute - izidakamizwa "Elefloks" (500 mg) esithathwayo nsuku zonke izinsuku eziyishumi noma amasonto amabili;
  • umphakathi-atholwe inyumoniya - usebenzisa 1000 mg izidakamizwa ngosuku e 2 ngemithamo ahlukaniswe amasonto 1-2;
  • nzima ukutheleleka, ezithinta ngomgudu womchamo - umthamo nsuku zonke oluhambisana 250 mg zomuthi, ubude course kancane isikhathi esingaphezu kwesonto, ukuphathwa kungapheli, uma kunesidingo;
  • zokugula, esithinta ngomgudu womchamo, futhi azikho izinkinga ezingase zivele - mayelana 4 izinsuku wamukelwa 250 mg zomuthi;
  • prostatitis ezibangelwa amagciwane, - zidinga ukwelashwa eside, ngezinye izikhathi phakathi kwezinsuku ezingu-28 ngo-500 mg "Elefloksa" usuku ngalunye;
  • sinusitis - Ukwelashwa ukukhiqiza izibhebhe umthamo zonke izinsuku we mg 500;
  • izifo intraabdominal - umthamo ekuphathweni nsuku zonke 500 mg, ubude Yiqiniso ekwelapheni eziyinkimbinkimbi - amasonto 1-2;
  • izifo lapho isikhumba ethintekile kanye ezithambile izicubu - yokwelapha isidingo nge double ethola 250 mg noma 500 mg izidakamizwa nsuku zonke amasonto amabili;
  • sofuba amelana isenzo nezinye izidakamizwa - ukuze bayothola ukwelashwa eziyinkimbinkimbi kuyadingeka ukuthatha nsuku zonke mg 500 izidakamizwa (bangathola up 2-emhlanjini) izinyanga ezintathu.

Iziguli isifo sezinso ngaphansi ezithile ukubaluleka QC (ml / iminithi) "Elefloks" yokusetshenziswa bangathola kanje:

  • QC 50-20 - lokuqala ukuthatha 250 mg, futhi kamuva - 125-250 mg (mhlawumbe ahlukaniselwe izikhathi eziningana);
  • QC 10-19 - lokuqala ethola 500 mg ngelanga, nge okunye ukwelashwa - 125 mg ngayinye amahora 12-48;
  • CC ngezansi 10 - wonke umuntu wenza okufanayo njengoba kwenzeka langaphambilini, kodwa imithi isetshenziswa okungaphezu kokukodwa amahora 12-48, kuthi njalo ngemva kwezinsuku 1-2.

Yenziwe isixazululo "Elefloks" weThrojani ukubeka okungenani ihora. okunye ukwelashwa incike isimo lesiguli. A shintsho amaphilisi ukuze umthamo, okuyinto ubeke weThrojani. Kulezo zimo lapho umzimba womuntu wayeyizwa zelashwe peritoneal futhi hemodialysis esasikhipha ngemithamo ezingeziwe nomuthi liyadingeka.

Ukwelashwa ezigulini esezikhulile abanezinkinga isibindi, kwenziwe amahora 48-72 noma ngaphezulu, kuze izimpawu zinyamalale, futhi ukubhujiswa okuphelele kwalelizwe Amagciwane.

Uma umthamo ukuthi uphuthelwe imithi njalo umthamo olandelayo iqondiswa noma kuthathwe ngokushesha ngangokunokwenzeka, ngalesosikhathi sebenzisa lwemithi ukukhwezwa.

Side Effects "Elefloks" izidakamizwa

"Levofloxacin" ( "Elefloks") kungacupha ukuthuthukiswa amathuba okuba nemiphumela engemihle. Phakathi kungenzeka ukusabela ezingezinhle zomzimba - ukubukeka dysbiosis, isifo sokusha kwesibindi kohlobo anobuthi, enterocolitis, dyspepsia. Kwangathi khona ubuhlungu bemisipha, ubuhlungu besisu, ikhanda elibuhlungu, uhudo, amajaqamba, ukundindizela, izinga lokushisa. Lapho ukusabela okungekuhle kuya izidakamizwa e-enzyme isibindi, umsebenzi kunyuke kungabonakala nasemkhakheni. Phezu ukuthola ezifana side effects njengoba nesifo pseudomembranous, okunye ukwelashwa, kusuka kube nzima.

Umuthi ngezinye izikhathi kuhambisana discoordination lapho wenza ukunyakaza, khona lability ngokomzwelo, ukucindezeleka nezinkinga ukulala. Kwezinye izimo, kubonakala thuthuva ukwazi, lokuhogela ukunambitheka. Ukuze uhlu ukusabela ezingezinhle zihlanganisa arthralgia, thrombocytopenia. Kwangathi ukuthuthukisa kahle agranulocytosis, paresthesia. Isiguli Kungaletha leukopenia, eosinophilia.

Ngokuphathelene nezinye imiphumela emibi ngesikhatsi ukwelashwa "Elefloks" ejenti kuhlanganisa yokusetshenziswa syndrome asthenic, kahle kungakhuphula izinga likashukela, imfiva, porphyria acute isesimweni, isifiso sokudla kakhulu, tachycardia, arrhythmia futhi ukwehla okukhulu komfutho wegazi (kukhona kungenzeka kokuwa).

Ngezinye izikhathi kukhona komzimba nezinto, lapho evuthayo futhi ukulunywa kwesikhumba, ukuthuthumela yezingalo nemilenze. Okungenzeka ukutheleleka yesibili. Kungenzeka ukubukeka photosensitivity, peripheral. Ukuthola yini imiphumela emibi - isizathu ukwelashwa kudokotela.

Overdose "Elefloksa"

Njengoba lingekho ikhambi, ukweqisa izidakamizwa yokwelapha lingaze kudinga. Phakathi izindlela eziphumelelayo ukuqeda isimo esinjalo - zelashwe peritoneal, hemodialysis.

Izixwayiso

Iziguli abasele emva kokwelashwa kusho ukubika "Elefloks" impendulo ukusetshenziswa ngokucophelela imithi ezimweni ezithile. Ezinye iziguli adinga kweso lwezokwelapha saziso.

Nge ukunyamalala umzimba okusezingeni eliphezulu lokushisa izinkomba yokwelapha kumele waqhubeka izinsuku 2-3. Ukwelashwa kakhulu nenyumoniya esilazayo kudinga ukusetshenziswa kwezidakamizwa eziningi, ngaphandle kwalokho elamukelekile engashiywa.

Phakathi ukwelashwa kufanele bakugweme kakhulu ukuchayeka kubo elangeni futhi yokufakelwa UV ukukhanya ngenxa ingozi photosensitivity.

Kukhona neminye imininingwane ezidinga ukunakwa. Noma yiziphi izinguquko empilweni kufanele wazise udokotela wakho.

Inhlanganisela "Elefloks" izidakamizwa nezinye izidakamizwa

Hlanganyela kunemithi noma amaphilisi owaphuzayo, "Elefloks" sithuthukisa noma kunciphisa ithonya lazo. Kungenzeka okufanayo nge isenzo izidakamizwa. Uma kunesidingo, ukuphathwa nezinye izidakamizwa esikhathini ukwelashwa "Elefloksom" Kufanele uqaphele ukuthi bangase bangakwazi ehambisanayo. Noma yiziphi izinguquko eziphathelene imithi, kufanele kuxoxwe nodokotela wakho.

"Elefloksa" Izindleko

Kuye ifomu Isikali "Elefloks" intengo izidakamizwa ruble mayelana 760-940. amaphilisi ngendlela umthamo mg 500 (№ 10). Mayelana 345-450 ruble. Kuyinto isixazululo emthanjeni (100 ml).

Izibuyekezo sokulungiselela "Elefloks"

Ngokuvamile, iziguli omuhle sebuhlaziyiwe izidakamizwa. Ngokusho kwabo, "Elefloks" ezisheshayo futhi kwenza kube nokwenzeka ukwelapha izifo eziningi omsakazo ezithathelwanayo.

Umuthi ngokuvamile iqondiswa iziguli ukulwa ngamagciwane eziningana izimo zokucabanga okubangelwa isifo uma kunesidingo.

Kwesobunxele emva kokwelashwa kusho "Elefloks" izimpendulo ibonisa izenzeko ezingavamile ukusabela ezingezinhle. Imiphumela engemihle ngokuvamile simnene futhi zinyamalale ngokuphelele lapho ukwelashwa usuphothuliwe.

Analogs "Elefloks" izidakamizwa

Izidakamizwa kabani isinyathelo kufana ukuthi kuhlinzekwe emzimbeni "Elefloks", zikhona ngamanani amakhulu. Asikwazi ukuhlukanisa izidakamizwa ezifana "Maklevo", "Leobeg", "Lebel". Azi kungenzeka ukusetshenziswa njengendlela esikhundleni "Lefoktsina", "Levofloxacin", "Glewe", "Ivatsina". Lezi zimali zibhekene ngqo okuvame kakhulu kanti zisetshenziswa eyolanda Analogue emuthini "Elefloks" uma kudingekile. Inani analogue ngezansi, umphumela ukusetshenziswa kwabo kufana.

"Elefloks" libhekisela izidakamizwa sina futhi kungabangela eziningi engemihle. Ngaphambi ukusebenzisa, kubalulekile ukufunda ngokucophelela imiyalelo. Ukusetshenziswa Its for ekwelapheni kufanele sigcwaliswe kuphela ngemva kudokotela, okuzokwenza ukulandela izinguquko ezenzeka emzimbeni.

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