ImpiloAmalungiselelo

Drotaverina hydrochloride

Drotaverina hydrochloride iphathelene izingoma ezithaka imithi ukuba umphumela spasmolytic. umsebenzi wayo siqondiswe imisipha abushelelezi wokugaya ukudla izitho, urogenital futhi biliary uhlelo, kanye semithambo bushelelezi imisipha ungqimba. Drotaverina hydrochloride (Nospanum), benemihelo ka bushelelezi imisipha izingqimba, uyakwazi ukuqeda cramping. Ngaphezu kwalokho, izidakamizwa kuthuthukisa izicubu umsoco umoya-mpilo: ukhulisa mafutha anciphisa isikhala esingaphakathi semithambo. Drotaverina hydrochloride unekhono ukushintsha of cell ulwelwesi ezingaba futhi permeability. I nomuthi kunciphisa umsebenzi enzymatic of phosphodiesterase, ikhuthaza uhambisane (iyunifomu) ukwandisa amazinga ekamu futhi ukumuncwa kokuqala kwe-calcium ion cells.

Drotaverina hydrochloride elinesimo ophansi kokubonisa ne-plasma amaprotheni. Isikhathi esiningi ke sibopha ukuthi beta-alpha-globulin,-albumin. Kungakapheli nemizuzu engamashumi amane nanhlanu, futhi ayisithupha ngemva kokuphathwa ngomlomo isicelo plasma ububonisa lokuhlushwa isiqongo we ketshezi esebenzayo. Ingxenye-ukuphila oda amahora amabili nambili. Excretion of metabolites ekhiqizwa ngokuyinhloko umchamo. Ingxenye excretion zomuthi kwenzeka indle.

Nomuthi (ngesimo umjovo, kanye amaphilisi) inikezwa ukuqeda izinhlungu uhlamvu spastic cupping spasm. Drotaverina hydrochloride ikhombisa isilonda esiswini, cholecystitis, ukuqunjelwa, spastic omsakazo, pyloric bushelelezi imisipha spasm futhi cardinal esiswini ikhadi, cystitis, nephrolithiasis, proctitis, pyelitis futhi uretrolitiaze. Umuthi isetshenziswa amajaqamba emathunjini kubangelwa ukubambezeleka amagesi kanye nesifo spastic. I nomuthi angasetshenziswa lapho siqhuba ukuhlola, kuhlanganise holetsistografii. Drotaverine esiwabelwe vasodilatation ekuhlonzeni semithambo bushelelezi kwemisipha izinhlungu zibe ungqimba remover bekhanda spasm izitsha palsy. izidakamizwa ngokuvamile sisetshenziswa algodismenoree practice gynecological. I nomuthi uyakwazi ukuvimbela nekugwema bushelelezi imisipha amajaqamba kwesibeletho ngesikhathi sokukhulelwa futhi esimweni okusongela isisu. Liphinde wabonisa esikhathini wokuthumela spasmolysis futhi eside ukuvezwa lesizalo emphinjeni kanye at izikhathi nangemuva kokuzalwa komntwana.

hydrochloride Drotaverina. Imiyalelo.

A ukulungiselela ngesimo amaphilisi ukuze uyiswe ngomlomo. Tablets akufanele ezokuhlafunwa noma afahlazekile, kumele wonke kugwinywe, ngamanzi eziningi ezanele. Umuthi akuxhomekile isikhathi ngemva kwesidlo. Umthamo kanye isikhathi sokwelashwa kunqunywa ngamunye by udokotela ukuba khona.

Intsha (phezu ibe neminyaka eyishumi nambili) kanye nabantu abadala ukuze akhulule izinhlungu spastic ukhethe 1-2 amaphilisi (40-80 mg) izikhathi ezimbili noma ezintathu ngosuku.

Izingane ezingaphansi kweminyaka eyishumi nambili sokulungiselela kunikezwa ngokuhambisana aphoyintimenti udokotela.

I nomuthi ngesimo umjovo iqondiswa intramuscularly. Ezigulini ezine-esingamahlalakhona kwezinso noma hepatic, kungase kukwenze wephuze ukwethulwa izidakamizwa ngemithambo yegazi. Le ndlela isebenza kuphela emva Ukwamukelwa evundlile isiguli. Ngo-peripheral ukuphazamiseka kwegazi lapho kubangelwa semithambo imisipha bushelelezi spasm ungqimba kube kancane ekuphathweni intraarterial.

Njengomthetho, iziguli ukubekezelela imithi. Nokho, kwezinye izimo, kungase kube khona emibi. Ngokwesibonelo, iziguli zingase zibhekane isicanucanu, sezinyawo kahle, ukuhlanza. Kungenzeka, futhi CNS neziyaluyalu, ezifana ukwephulwa eziningi ulokhu uphaphama futhi imodi ukuphumula (ubuthongo), ikhanda, yokufikelwa. Kwakukhona amacala iziyaluyalu esimiso senhliziyo nemithambo yegazi, owabonakaliswa tachycardia, arrhythmias, ukwehlisa ingcindezi. Libuye ukuvuvukala okungenzeka le mucosa acinene, komzimba nezinto, bronchospasm.

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