Impilo, Amalungiselelo
Tioktatsid®: analogue. Tioktatsid®: imfundo, intengo, ukubuyekezwa
Tioktatsid® - ukulungiselela thioctic (njengoba ibizwa-alpha-lipoic acid). Alpha-lipoic acid - antioxidant enamandla, kuyingxenye ebalulekile eyingozi eziningi kwamakhemikhali nezinqubo bokuphila emzimbeni womuntu, okuyinto ngaphansi kwezimo ezivamile futhi kukhiqizwa. Thioctic acid umsebenzi ukuvikela amangqamuzana omzimba emiphumeleni elimazayo radicals khulula. Ngaphezu kwalokho, thioctic acid kuyahluka umsebenzi detoxication futhi ehilelekile ukubuyiselwa endogenous uhlelo antioxidant emzimbeni. Ikakhulukazi, i-alpha-lipoic acid kuvusa sokubuyiselwa vitamin C no-E, coenzyme Q10, okwandisa lokuhlushwa glutathione antioxidant yangaphakathi.
Tioktatsid® kokuba umsebenzi nootropic, uvikele isibindi, kunciphisa lokuhlushwa igazi lipids, kuhlanganise i-cholesterol, kuvusa glucose ukusetshenziswa by kwezicubu zomzimba, lokho kukunciphisa ngokuphawulekayo ukudleka ezingeni layo egazini. Waba yini umphumela wesibindi ukwehla onjalo eziyinkimbinkimbi ithonya kuwukubonakaliswa insulin emzimbeni. Tioktatsid® futhi kunciphisa indlala, kuvusa okisleniyae acid okunamafutha, kanjalo uvimbele ukudala ezinye ekuqongeleleni fat umzimba kanye nekufaka ligalelo ukuzinza esisindo, kuhlanganise nokwelashwa ukukhuluphala.
Tioktatsid® BV (okusheshayo ukukhululwa) - umuthi ngezilinganiso uhlobo oluthile elungiselelwe ukuze athathe ke ngomlomo. umumo esinjalo siqinisekisa ukuthi umzimba uyokwenza ethile thioctic acid, ezingeni yayo plasma uzinze. Ngaphezu kwalokho, ukukhululwa ifomu okusheshayo ihlinzeka bioavailability okusezingeni eliphezulu we ketshezi esebenzayo.
I pharmacokinetics zomuthi Tioktatsid®
Ngenxa mkhakha okhethekile ukukhululwa esheshayo, wathola umzimba-alpha lipoic acid esifitshane imizuzu 15-20 of, egxile ngokuphelele ku igazi kokuqala ipheshana wokugaya ukudla. Kufanele kukhunjulwe ukuthi reception kanyekanye Tioktatsid® BV ngokudla kakhulu kuthinta ukumuncwa isithako esisebenzayo (alpha-lipoic acid). Ukuhambisana izincomo yokwamukela izidakamizwa - yokwamukela esiswini esingenalutho isigamu sehora ngaphambi kokudla - ukuvimbela ukuxhumana engadingeki nge ukudla, kulesi simo, inqubo ukumuncwa kwe-alpha-lipoic acid egazini ngesikhathi sakusihlwa, usuphethiwe. okuhlushwa enkulu yama thioctic acid plasma ifinyelela imizuzu engu-30 ngemva izidakamizwa isidlulile, kuba 4 UG / ml, lapho acid-alpha-lipoic, libhekene umphumela "pass lokuqala" ngokusebenzisa isibindi. I bioavailability alpha-lipoic acid reception Tioktatsid® BV ekwakhiweni kuyinto 85%. Izindlela eziyinhloko lokugayeka kokudla emzimbeni - namachibi futhi conjugation. Kufika ku-90% we-thioctic acid kanye nemikhiqizo yayo umzimba iqedwe nge nezinso. Ingxenye-ukuphila imizuzu engu-25.
Izinkomba polyneuropathy sikashukela kanye utshwala
Thioctic acid likhona impatho esezingeni lezi zifo ezilandelayo: peripheral ezihambisana systemic zezinzwa izifo izicubu. Radiculopathy. Parkinson. Stroke. Okunobuthi-hepatitis A no-C imnene kobukhulu ngokulinganisela. retinopathy sikashukela kanye edema macular.
Izimo izidakamizwa Tioktatsid®
Kuze kube manje akukho idatha okunokwethenjelwa ngokuphathelene umphumela isidakamizwa isidumbu sowesifazane phakathi nokukhulelwa kanye lactation, ukuze iziguli ezinjalo Tioktatsid® ayizange inikezwe. Ngesizathu esifanayo it is hhayi Kunconywa ukusebenzisa izidakamizwa ekwelapheni iziguli kabani yobudala engaphansi kuka-18 ubudala. Hypersensitivity ukuze imibuso eyakha lo izidakamizwa nakho contraindicated.
Isicelo, umthamo we izidakamizwa Tioktatsid®
I umthamo wansuku zonke lapho udle 600 mg zomuthi (eziqukethwe iphilisi elilodwa). Thatha imithi ngokuqinile esiswini esingenalutho, isigamu sehora ngaphambi kokudla kwasekuseni. I-Tablet kugwinyiwe lonke ngaphandle ukuhlafuna, ukugeza phansi ngamanzi. Uma kwenzeka kuba nzima, asetshenziselwa ukwelapha Tioktatsid® 600T senzelwe abaphathi emthanjeni. Nsuku zonke isiguli iqondiswa okuqukethwe kancane emthanjeni elilodwa isitsha (600 mg). Ukwelashwa Uthatha amasonto amabili kuya ngenyanga, bese wenza sibonane translation nesineke Tioktatsid® BV. Ukuvimbela ukusabela ezingafuneki eMbusweni isipetu ukuba iphathwe isixazululo okungenani 12 imiz.
Njengoba wenza izidakamizwa ingxenye ukuzwela ezahlukene ukukhanya, izitsha eziyisikhombisa asuswe ibhokisi ngokushesha ngaphambi izidakamizwa abaphathi. Okulandelayo, isiguli idluliselwe yokwelapha izidakamizwa Tioktatsid® DB 600 e umthamo 1 ithebhulethi ngosuku.
imiphumela emibi izidakamizwa Tioktatsid®
On the ingxenye pheshana emathunjini ngokuvamile ngokuthi isicanucanu. Okunye kuwukubonakaliswa ukungakhululeki phezu ingxenye isimiso sokugaya ukudla bungene - ukuhlanza, ubuhlungu Iwumbono esiswini namathumbu, izigqiki okuxekethile, ushintsho ukunambitheka - ukhathazekile, ezimweni ezingajwayelekile kakhulu.
komzimba (isikhumba ukulunywa, ukuqubuka emzimbeni, isifuba ukushaqeka anaphylactic) akuvamile uhlupho.
Kusukela isimiso sezinzwa kungenzeka ukhathazekile isiyezi.
Jikelele: ezimweni ezingajwayelekile kakhulu, ngenxa ezishukumisayo glucose kulahlwa izinqubo kungaba izimpawu wayephambanisa ka kahle kungakhuphula izinga likashukela (umbono anyakaza, ukujuluka, ikhanda elibuhlungu, ukudideka), okuyizinto umphumela ukwehla kwamazinga igazi glucose.
Tioktatsid® izidakamizwa ekuxhumaneni nezinye izidakamizwa
Uma izidakamizwa isetshenziswa kanye cisplatin, cisplatin attenuated.
Njengoba thioctic acid, aqukethe Tioktatsid® BV Tioktatsid® 600T ukhuthaza metal ngibopha is hhayi Kunconywa kanyekanye nensimbi amalungiselelo. Isikhawu phakathi reception Tioktatsida® nensimbi amalungiselelo, i-calcium, umlingo kufanele okungenani amahora ama-2. Ezimweni lapho Tioktatsid® isicelo kanyekanye ne temlomo ejenti hypoglycemic noma se-insulin, umphumela hypoglycemic kwala magciwane zingavela evelele. Kuyadingeka ukuqapha okuqukethwe glucose egazini, ikakhulukazi esigabeni sokuqala ukwelashwa.
Izixwayiso
A ukulungiselela amaphilisi is hhayi obala ukuze ukukhanya kuze ukusetshenziswa ngqo. Phakathi ukwelashwa kufanele uhlukane nale ukusetshenziswa ethanol, njengoba yokugcina kungenzeka kunomthelela ukuthuthukiswa polyneuropathy.
Analogue, intengo, ukubuyekezwa mayelana izidakamizwa Tioktatsid®
Tioktatsid® ukubaluleka ngesimo ampoules kuyinto ruble 1500 ngesimo amaphilisi -. Ruble 1700-3200. Okuzuzisa kakhulu emaphaketheni - amaphilisi 100 izinyanga ezintathu.
Tioktatsid® - namuhla kuphela izidakamizwa kokuba okusheshayo ukukhululwa ifomu esihlinzeka ukumuncwa esiphezulu lomcebo asebenzayo umzimba.
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