Impilo, Amalungiselelo
Medicine "Tiolepta": yokusetshenziswa, analogue, intengo, kanye nokubuyekeza of the ukulungiselela
Kungani sidinga umuthi "Tiolepta"? ekusetshenzisweni lo mhlahlandlela imithi izokwethulwa mathiriyeli lo sihloko. Ngaphezu kwalokho, kuwo uzofunda amafomu lapho izidakamizwa ikhishwe phambi kwethu, eminye ingxenye yalo, uma unazo contraindications side effects, kanye ukuthi kubiza malini futhi lokho kungenziwa indawo.
Khipha izinhlobo imithi ngezithako zawo
Ngayiphi fomu akhangiswe imithi "Tiolepta"? Okwamanje izidakamizwa itholakala amafomu ezimbili ezihlukene, okuyilezi:
- Ngo amaphilisi, camera aphuzi. Njengoba uhlobo esebenzayo izidakamizwa ukulungiselela iqukethe thioctic acid. nomuthi sihlanganisa asizayo izakhi. Bahlanganisa amazambane isitashi, aerosil A-300 (noma colloidal Silicon dioxide), microcrystalline cellulose, primelloza (noma i-sodium croscarmellose), ubisi noshukela (noma i-lactose), i-polyethylene glycol-400 (noma macrogol-400), uwoyela ocolisekileyo, i-calcium stearate, titanium dioxide, methylcellulose hydroxypropyl, quinoline ophuzi, polyethylene glycol-6000 (noma okuthiwa macrogol-6000), yellow yensimbi oxide. Ngo elinye ibhokisi kungaba 10, 60, 30 noma 90 amaphilisi.
- Ikhambi for ukumnika. Njengoba ketshezi esebenzayo, lolu hlobo nomuthi iqukethe thioctic acid. Njengoba for nye izakhi, lezi zihlanganisa meglumine, povidone, macrogol, namanzi umjovo. Umuthi itholakale emakhemisi ngo amabhodlela 50 no-25 ml.
I izakhiwo kwemithi sedivayisi yezokwelapha
Uyini izidakamizwa "Tiolepta"? Iziyalezo yokusetshenziswa Lithi kuyinto -ejenti umzimba. isithako wayo (i-alpha-lipoic acid) kuyinto antioxidant endogenous, okuyinto sibopha mahhala radicals.
kwakhiwa Thioctic acid is emzimbeni womuntu e inqubo decarboxylation oxidative alpha-keto acid. I nomuthi kunciphisa igazi glucose glycogen anda ivolumu isibindi. Ngaphezu kwalokho, lo izidakamizwa kalula unqobe insulin.
Ngokusho imiphumela yayo kwamakhemikhali izidakamizwa liseduze kakhulu amavithamini B Umuthi iye bahileleke ukulawulwa carbohydrate lipid umzimba. Ithuthukisa kokusebenza kwesibindi kudaleke exchange of cholesterol. Umuthi ungaba hypolipidemic, hepatoprotective, hypoglycemic nemiphumela ane-ukwehlisa.
Pharmacokinetics zomuthi
Emva kokuthola amaphilisi "Tiolepta" (600 noma 300 mg) ketshezi esebenzayo ku-ngokushesha futhi ngokuphelele ugxile kusukela ipheshana wokugaya ukudla. ukusetshenziswa ngesikhathi esisodwa ukudla kungaba kakhulu ukunciphisa ukumuncwa zomuthi. I bioavailability zomuthi ingu-30%. Umkhawulo igazi lokuhlushwa kufinyelelwe kumaminithi 40-60.
Lesi sidakamizwa ine umphumela ndima lokuqala ngokusebenzisa isibindi. Metabolites imiswe phakathi conjugation kanye namachibi ka ohlangothini chain.
Kuboniswa izidakamizwa umchamo (80-90%).
Izinkomba ngokusetshenziswa idivayisi yezokwelapha
Kwezinye izimo, prescribers "Tiolepta"? Yokusetshenziswa iqukethe uhlu elandelayo ukufundwa:
- polyneuropathy utshwala;
- polyneuropathy sikashukela.
Izimo ukusetshenziswa idivayisi yezokwelapha
Uma ungeke ukwazi ukusebenzisa i- izidakamizwa "Tiolepta"? Yokusetshenziswa kwaleli thuluzi ikhombisa Izimo ezilandelayo:
- isikhathi sokukhulelwa;
- Wezingane yobudala (ukuphepha nokusebenza ngempumelelo zomuthi engakaze isungulwe);
- Phakathi ibele ingane (akukho isipiliyoni esanele izimali);
- Owengeziwe nesineke kuvelana izidakamizwa.
Indlela ukuthatha imithi "Tiolepta 600"?
Yokusetshenziswa kwe-ithuluzi inikeza ukuthi izidakamizwa ngesimo amaphilisi ngokuvamile ezinqunyiwe imizuzu engu-30 ngaphambi kokuba kudliwe lokuqala (isb ngaphambi kokudla kwasekuseni). I nomuthi kufanele kuqashelwe imali mg 600 kanye ngosuku. Tablets akufanele ezokuhlafunwa. Kufanele wageza phansi ngamanzi amancane. Isikhathi inkambo ukwelashwa kufanele azimisele kuphela udokotela ukuba khona.
Ngo amafomu kakhulu izifo ezifana polyneuropathy sikashukela kanye utshwala, izidakamizwa esebenzayo iqondiswa ngemithambo yegazi (iconsa kuphela). I nomuthi iqondiswa emqulwini ka 50 ml kanye ngosuku. Ekuqaleni yokwelapha Yiqiniso izidakamizwa iqondiswa ngemithambo yegazi phezu amasonto 2-4. Ngemva kwalokho, ushintsho ukuze yetemlomo zomuthi at umthamo 300-600 mg ngosuku. Isixazululo for umjovo kufanele sinikezwe kancane (hhayi ngaphezulu kuka-50 mg isithako esisebenzayo ngomzuzu).
Izidakamizwa ukweqisa izidakamizwa (izimpawu, ukwelashwa)
Kwenzekani uma ungenawo ukulandela izincomo udokotela athathe umthamo enkulu izidakamizwa "Tiolepta"? ochwepheshe lezivakashi bathi izimpawu ezilandelayo ukweqisa izidakamizwa kungenzeka kulokhu, isicanucanu, ukuphathwa ikhanda, ukuhlanza. Indlela esiphatha ngayo isiguli ezimeni izidakamizwa ukweqisa izidakamizwa "Tiolepta"? Kufanele ukuchitha yokwelapha lingaze.
Imiphumela emibi ngemva kwesicelo se-nomuthi
Ngokuvamile, lesi sidakamizwa "Tiolepta", intengo olubonakaliswa kancane ibekezelelwe aphila kahle. Nokho, kwezinye izimo? Kuvelelani ohlangothini imiphumela elandelayo:
- ipheshana wokugaya ukudla: ukuqunjelwa, isilungulela, ukuhlanza kanye nesicanucanu.
- Yokungezwani komzimba: okunhlobonhlobo cutaneous (isb urticaria).
- Umzimba: kahle kungakhuphula izinga likashukela (ngenxa ngcono glucose abatholako).
Ukuxhumana nezinye izidakamizwa
Ngingakwazi ukusebenzisa umjovo noma amaphilisi "Tiolepta" nezinye izidakamizwa? Impendulo yalo mbuzo kufanele kube ukufunda kusukela ochwepheshe. Uma ungenayo i-kungenzeka esinjalo, sincoma ukuthi ngokucophelela ufunde imiyalelo enamathiselwe. Ngokusho lokhu ukulungiselela, ikakhulukazi, thioctic acid, usabela kahle ionic metal izakhiwo. Kule ndaba, yokwamukela ngesikhathi esisodwa nomuthi kungaba kakhulu ukunciphisa ukusebenza kwe cisplatin.
Ukuba nomuthi "Tiolepta" ekuseni ukusetshenziswa amalungiselelo magnesium nensimbi futhi uqede imikhiqizo yobisi (ngenxa okuqukethwe kwe-calcium) kumele kube ntambama noma ebusuku. Ukusetshenziswa ngesikhathi esisodwa nomuthi kalula ukuthuthukisa umphumela we-insulin kanye kwezidakamizwa temlomo hypoglycemic. Asinakusho ukuthi i-ethanol iyehlisa umsebenzi oqabulayo-alpha-lipoic acid.
isiqondiso Specific on ukusetshenziswa idivayisi yezokwelapha
Labo ezigulini thatha izidakamizwa "Tiolepta", isikhathi sokwelashwa kufanele uyeke ukuphuza uphuzo utshwala.
Njengoba for iziguli sikashukela, inkathi ukwelashwa kudinga ukuqapha njalo. Lezi ziguli badinga hlola lokuhlushwa glucose egazini. Ikakhulukazi kubalulekile ukwenza esigabeni sokuqala ukwelashwa. Kwezinye izimo kubalulekile ukunciphisa umthamo we-insulin noma ama-ejenti temlomo hypoglycemic. Lokhu kuyadingeka ukuze ugweme kahle kungakhuphula izinga likashukela.
Umuthi 'Tiolepta ": nozakwabo futhi izindleko imithi
Ukulandela aphoyintimenti isiguli umuthi ngokuvamile nesithakazelo umbuzo kubiza malini. Okwamanje, le imithi angathengwa at ezahlukene amanani. It akuxhomekile nje kuphela esimweni ethile ekhemisi iketango eziseceleni ezimpahleni, kodwa futhi ukuma ukukhululwa zomuthi kanye ubuningi iphakethe.
Ngakho-ke yini izindleko imithi "Tiolepta"? Intengo zomuthi kuyahlukahluka 600-700 ruble Russian 30 Tablets (600 mg). Uma udinga umthamo ezincane, bese ukuthenga esilinganayo izidakamizwa kungabangwa ruble 300-400 (300 mg).
Manje ngoba sewuyazi ukuthi kungakanani isikhungo sokwelapha "Tiolepta 600". Intengo yaleli izidakamizwa impela high. Kuyinto leli qiniso odlulela iziguli eziningi esikhundleni izidakamizwa ne analogue eshibhile. Lezi zihlanganisa imithi ezilandelayo: "Lipoic acid", "Neyrolipon", "Lipotiokson", "Oktolipen" kanjalonjalo.
Yini okunye esikhundleni imithi "Tiolepta"? Analogue kwaleli thuluzi kungaba ushibhile nje kuphela kodwa futhi kuyabiza ngaphezu original. Le mithi ihlanganisa lokhu okulandelayo: "Alpha-lipoic acid", "Lipamid", "Beplition", "thioctic acid," "Thiogamma", "Tiolipon", "Thioctacid", "Espa-lipon" et al.
Kufanele kuqashelwe ukuthi esikhundleni analogue of kadokotela, "Tiolepta" kufanele kube abanolwazi professional. Lokhu kungenxa yokuthi la izidakamizwa angase abe ezahlukene ngokuphelele imiphumela eminingi engemihle njengezindlela contraindications umthamo.
isitoreji Izindlela
Gcina izidakamizwa "Tiolepta" kufanele kuphela endaweni epholile futhi amnyama, nalapho kungekho ukufinyelela izingane ezincane. Impilo eshalofini zomuthi emibili ngenxa amaphilisi kanye isixazululo iminyaka emithathu.
Ukubuyekeza ku imithi
Yini iziguli uthi ngemithi enjalo, njengoba "Tiolepta"? Izibuyekezo lokhu ukulungiselela akhayo ngokwezinga elikhulu. Ngokusho iziguli, le nomuthi "Tiolepta" limelela ithuluzi elikahle kakhulu ubuhlungu emuva futhi emikhawulweni aphansi. Umbhali wayevame ukunezela lokhu izidakamizwa elibekelwe iziguli ngemva kokuhlinzwa in iziguli ngifundise ngesifo sikashukela. Leli thuluzi kahle ukuze uthole ezinyaweni zakhe, njengoba u-40% iziguli sikashukela, kukhona izifo nezinzwa neuropathy.
Medicine "Tiolepta" kusiza ukuthi uyoqeda ubuhlungu futhi ekudambiseni isimo iziguli, ikakhulukazi uma ukhuluphele.
Asinakusho ukuthi lokhu izidakamizwa ngokuvamile ebekiwe njengendlela yokukwenza inhlanganisela isibindi sibe sesomile.
Ngokuqondene Izibuyekezo ezingezinhle ke lesi sidakamizwa "Tiolepta" ayatholakala. Ezimweni eziningi ezihlobene yokuthi ngemuva kokusebenzisa ithebhulethi noma komjovo izixazululo iziguli ziba nemiphumela emibi ezifana isicanucanu, ukuhlanza kanye isilungulela ezinzima. Ngaphezu kwalokho, ezinye iziguli zithi izidakamizwa akukuniki yimuphi umphumela. Ngenxa yalokho, iziguli kwaphoqeleka ukuthi kubhekisiswe futhi ukufinyelela ubuciko, abelwe kubo ngendlela efanele kwezidakamizwa.
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