ImpiloAmalungiselelo

"Desloratadine": yokusetshenziswa, nozakwabo yangempela

komzimba kwenzeka kuphela kubantu abanegciwane hypersensitive izivikeli mzimba. Ngokuvamile, lapho zenzeka nge okuphindaphindiwe allergen ukuchayeka emzimbeni, ngaphambili batiswe kubo. Izimo ezinjalo ngokuvamile kuvinjelwe umuntu nokuphila okuvamile.

Ukuze basize iziguli nge izinhlelo hypersensitive mzimba, weenhlahla eseqala ukuveza ekhethekile elwa ne-iguliswa, okuyinto kakhulu ngcono izinga lempilo kanye isimo lesiguli.

Izindlela ethandwa kakhulu okuhloswe ngazo ekulweni ukubonakaliswa nomzimba, buyisidakamizwa "desloratadine". Iziyalezo ukusetshenziswa analogue, ifomu ukukhululwa kanye nobufakazi lomutsi izokwethulwa ngezansi.

Incazelo, emabhokisini ifomu ukukhululwa kanye nokusungulwa

I nomuthi "desloratadine", yokusetshenziswa okuyinto ibekwe inqwaba amakhadibhodi, ekhiqizwa ngesimo amaphilisi round blue kanye namafomu biconvex. Ziyakwazi ifilimu-camera futhi ube core emhlophe (esigabeni cross).

Isithako asebenzayo lokhu ejenti kuyinto desloratadine. Ngaphandle-ke, lichaza ekwakheni amaphilisi kanye zihlanganisa izakhi ezengeziwe ngesimo corn isitashi, calcium hydrogen phosphate dihydrate, microcrystalline cellulose, magnesium stearate futhi talc.

Ngokuphathelene ifilimu enamathela, esenziwe ingxube dry ehlanganisa polyvinyl utshwala, ama-titanium dioxide, talc, makragola 3350, Aluminium lacquer udayi futhi ephuzi yensimbi oxide.

Thenga imithi angabhekwa ku amaphakheji uhlaka kanye amakhadibhodi amabhokisi, ngokulandelana.

pharmacodynamics zomuthi

Kuyini umenzeli antiallergic ezifana "desloratadine" (amaphilisi)? Yokusetshenziswa ibonisa ukuthi lokhu blocker N1- histamine yokwamukela, okuyinto kunomphumela nehlala njalo.

Lokhu nomuthi oyibamba metabolite ka loratadine. Ngo potency kwalo oludlula ke ezikhathini 2-4.

izidakamizwa Okubukwe ekuvimbeleni uchungechunge ukusabela ukuvuvukala nomzimba (Ukukhululwa cytokines, chemokines, interleukin futhi prostaglandin D2).

Yokungezwani komzimba amaphilisi "desloratadine" babe decongestant nomphumela antipruritic, wenze kube lula komzimba, ukunciphisa hyperreactivity bronchial, futhi allergen eqondene ukubonakaliswa bronchospasm, kanye ukuqeda izinhlungu zibe of imisipha abushelelezi. Umthelela izidakamizwa, ezithathwe ngomlomo, siyenzeka usuku lonke.

Kumele kuqashelwe futhi ukuthi izidakamizwa akunamthelela le CNS, kufaka phakathi umthamo 7.5 mg. Akanawo imiphumela cardiotoxic, umthelela ijubane lengqondo ukusabela ukupholisa.

izici kinetic

Lapho ukumuncwa lesi sidakamizwa "desloratadine"? Yokusetshenziswa ubonisa ukuthi ukumuncwa zomuthi kusukela ipheshana emathunjini wenziwa.

Ubuningi aphansi zomuthi atholakala igazi emva kwemizuzu 35, kanye elikhulu - emva 3 h.

I asebenzayo izidakamizwa ketshezi kuyinto 87% eboshiwe plasma amaprotheni. I wathola kungakapheli amasonto amabili ngesikhathi umthamo mg 20 ungakuvumeli ukuba ukubukeka izimpawu cumulation.

Ukudla ukudla akunamthelela ukusatshalaliswa izidakamizwa abantu.

Kubhekwe yokukhalaza ngokushesha akheka. It ibonakala nge Inobulongwe nomchamo izidakamizwa ukuqedwa isigamu-ukuphila amahora 20-35.

izinkomba

Ngaphansi akukho kuwukubonakaliswa komzimba kufanele libekwe lesi sidakamizwa "Desloratadine Teva?" Yokusetshenziswa ukhombise izinkomba ezilandelayo:

  • urticaria ezingamahlalakhona;
  • hay fever;
  • unyaka wonke rhinitis iguliswa.

Izimo amaphilisi

Ngaphansi kwaziphi izimo asivunyelwe ukusebenzisa ithebhulethi "desloratadine"? Yokusetshenziswa (izingane lokhu izidakamizwa inikezwa kuphela abafinyelela eminyakeni yobudala engu-12) ibika ukuthi Izimo ezilandelayo izidakamizwa:

  • ngesikhathi sokukhulelwa;
  • anda kuvelana izithako zomuthi;
  • ibele;
  • zokungezwani ne-lactose;
  • malabsorption glucose-galactose.

Nomuthi "desloratadine": yokusetshenziswa

kufanele Ngithatha kanjani izindlela wathi? Ngokusho kochwepheshe, lokhu izidakamizwa kudinga ekuphathweni lolukhulunywako esifanayo.

Ukusetshenziswa amaphilisi kuzimele ukusetshenziswa ukudla. ithebhulethi Antiallergic ezokugwinywa lonke.

Izingane Ezisathomba engaphezu kwengu-12 ubudala kanye abadala imithi ezinqunyiwe umthamo 5 mg kanye ngelanga.

Mayelana emagama lafanako ezinjalo, njengoba "Desloratadine Teva", isetshenziswa esilinganayo kanye ne kaningi efanayo.

Isikhathi ukwelashwa ngaphansi ukucatshangelwa izindlela incike ukuvama ukuqala isifo nomzimba.

Njengoba wazi, ngesikhathi ngakanye izimpawu rhinitis kungenzeka esikhathini esingaphansi kwamasonto ezine ngonyaka. Ukwelashwa kwezifo ezifana kumele igcine kuphela emva ukunyamalala zonke izici zawo. Eqhubeka izidakamizwa lapho kuyinto efiselekayo kabusha zenzeka.

Kepha rhinitis ophikelelayo, izimpawu zalesi yokungezwani komzimba kungenzeka kanengi ukudlula amaviki 4 ngonyaka. Ngokuvamile, okuvela kuyo ukusabela okunjalo ngenxa ukuthintana njalo ne allergen. Ezimweni ezinjalo, ukwelashwa kufanele siqhubeke njengoba nje ukuxhumana allergen usuphothuliwe.

side effects

Noma yimuphi ukusabela ezingezinhle zenzeka seziguli ezithola amaphilisi "desloratadine"? Yokusetshenziswa, kumpendulo yekhasimende kubonisa lokhu okulandelayo side effects:

  • angnonevrotichesky edema, ikhanda elibuhlungu, anaphylaxis, ukusangana, ukuba nesiyezi, amajaqamba, ukulunywa, isiyezi, ukuqubuka, ukuqwasha, urticaria;
  • ukozela, tachycardia, lengqondo giperaktnviost, palpitations;
  • nomlomo owomile, myalgia, ubuhlungu besisu, ukukhathala, isicanucanu, umphimbo obuhlungu, ukuhlanza, dysmenorrhea, neuralgia;
  • umsebenzi kunyuke enzyme isibindi, uhudo, kukhuphuke bilirubin okuhlushwa, i-hepatitis.

amacala ukweqisa izidakamizwa

Kuzokwenzekani nge amazinga okukhishwa okwandisiwe izidakamizwa ukuthatha "Desloratadine Teva?" Ukufundiswa uthi ukusetshenziswa nsuku zonke izibhebhe 20 mg amasonto amabili akuzange kumenze yiziphi izinguquko CCC.

Kufanele kuphawulwe ukuthi reception we nomuthi ngezilinganiso of 45 mg izinsuku 10 awazange afake isandla prolongation qt isikhawu nokubukeka iyiphi enkulu engemihle.

izimali Okufanayo kanye nezindleko

Uma kukhona Izimo kuya "desloratadine" amaphilisi bangakwazi kuthathelwe indawo izindlela ezifana "AlergoMaks", "Erius", "Elisa", "Nalorius", "Lordestin", "Ezlor", "Des", "Eridez". Indlela isicelo izidakamizwa ezinjalo kungase kungafani indlela ekutholeni "desloratadine". Ngakho-ke, zimise kuphela Udokotela awe-aleji abanolwazi

Thenga imithi kungaba kucatshangelwe ruble 200-320 (amaphilisi 10).

Uphenyo ejenti antiallergic

Manje uyazi ukuthi imithi edingekayo "desloratadine". Yokusetshenziswa zomuthi seyenziwe ngenhla.

Lesi sidakamizwa kungokwalabo eziningi zalezi zinsuku futhi ethandwa antihistamine.

Iziguli bathi kuyaphumelela kakhulu ekwelapheni izifo nomzimba. A iphilisi ngokushesha aqede ukuminyana acinene.

Futhi kubhekwe nomuthi ngokuvamile isetshenziswa ngesikhathi esifanayo ne rhinitis somoya (atopic).

Abantu ne urticaria ezingamahlalakhona washeshe aqede zonke izimpawu zesifo.

Enye inzuzo yokuhamba kwesikebhe lo muthi ukuthi akanayo nemiphumela okulalisayo kanye nemiphumela omubi enhliziyweni.

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