Impilo, Amalungiselelo
"Artrokol" (gel): yokusetshenziswa, analogs kanye nokubuyekeza
kufanele ngisebenzisa kanjani izidakamizwa "Artrokol" (gel)? Yokusetshenziswa zomuthi uzobe achazwe kulo magazini. Futhi, uzofunda kulokho imithi enqunyiwe iziguli ukuthi unakho le analogue, futhi noma yikuphi ukuphawula ngalo eshiya umthengi.
Ukwakhiwa, izidakamizwa iphakeji ezakheke
"Artrokol '- gel (2.5%) ukusetshenziswa yangaphandle. Ngo ukudayiswa ufika kule aluminium tube 45 wayebuye ebhokisini amakhadibhodi kanye kwezidakamizwa manje Ipheshana nge imiyalelo enemininingwane ukusetshenziswa.
Lokho iqukethe izidakamizwa yangaphandle "Artrokol" (gel)? 100 g le ndlela yokuxhumana equkethwe 2.5 g isithako esebenzayo, njengoba ketoprofen. Ngaphezu kwalokho, e-izidakamizwa ngaphansi ukucatshangelwa ukusekelwa zici ezilandelayo: trolamine, Carbomer 980, 96% ethanol, amanzi ahlanzekile kanye methyl parahydroxybenzoate.
Umgomo we operation ye nomuthi
"Artrokol" - ijeli, isithako esebenzayo ketoprofen. Wathi nomuthi uphakathi kwabantu abangenalo leli izidakamizwa eqeda ukuvuvukala nonsteroidal, kanye nemikhiqizo ye arylpropionic acid.
nomuthi Base okunikezwe inikeza eqeda ukuvuvukala kanye analgesic umphumela, okuyinto eyenzeka ngesikhathi okusithiyayo non-ukukhetha Cox-1, bradykinin futhi Cox-2, kanye ulwelwesi njengoba sinjalo (lysosomal) kanye okusithiyayo of macrophage ukufuduka.
Ngaphezu kwalokho, izidakamizwa "Artrokol" (gel) liveza izindawo anti-inflammatory futhi ngizwa. It uyakwazi ukwenza phezu ekuseni khulu, ngemuva kwesikhathi cell isigaba semithambo we ukuvuvukala. Futhi, lolu izidakamizwa kubambezela platelet wokuhlanganisa.
Izimfanelo pharmacokinetic ka
Ngokusho imiyalelo enamathiselwe, ketoprofen (isithako esebenzayo ye nomuthi) emva isicelo nezokusigcoba isikhumba amuncwa umzimba, bese lingena singene maphakathi ukuvuvukala futhi ngesikhathi isikhathi eside egcina oyifunayo lokuhlushwa zokwelapha emisipheni.
Absorption zomuthi ku kwegazi incane (5% we umthamo esetshenziswa). Kulokhu, ukumuncwa lwalo emfudlaneni igazi kancanekancane.
I lokuhlushwa isithako zomuthi (usebenzisa 50-150 mg ketoprofen) egazini emva 7.5 amahora kuyinto mg 0.08-0.15 kuphela / ml.
Izidakamizwa "Artrokol" (gel) futhi injongo yaso?
I izinkomba for ukusetshenziswa ijeli olucutshungulwayo yilezi ezilandelayo uthi:
- myalgia, rheumatism kanye rheumatism umsuka;
- izifo of the system zemisipha (kuhlanganise i-rheumatoid arthritis, syndrome articular ngesikhathi exacerbation sifo, ankylosing spondylitis, arthritis psoriatic, osteochondrosis, i-osteoarthritis ka kwasendaweni ezahlukene, lesion sokuvuvukala imisipha, nemisipha, sciatica, bursitis noma lumbago);
- ingxenye ukwelashwa eyinkimbinkimbi ukuvuvukala pathologies emithanjeni (isib phlebitis, periphlebitis), izindlala zamanzi noma lymph (isib lymphangitis, lymphadenitis olukha phezulu);
- ukuvuvukala ukucindezeleka kwangemva kwenhlekelele of the system zemisipha kanye izicubu zomzimba ezithambile (kubandakanya nokwelashwa lingaze yokulimala ayinzima, kuhlanganise Ukwenyela, ukulimala ezemidlalo, Ukwenyela noma izinyembezi we imisipha kanye nemisipha, nemivimbo, ubuhlungu ukucindezeleka kwangemva kwenhlekelele).
Uvala ukusetshenziswa
Luthini olwakho "Artrokol" wamafutha kusiza, thina kuchaziwe ngenhla. Nokho, lokhu kusho ukuthi kukhona Izimo. Lezi zihlanganisa lokhu okulandelayo:
- yobudala engaphansi kwengu-12;
- sensitivity high izakhi zomuthi kanye acetylsalicylic acid nezinye ama-NSAID;
- senyanga yesithathu bekhulelwe nangenkathi bencelisa.
Izidakamizwa "Artrokol" (gel): yokusetshenziswa
Ukuze ekwelapheni ijeli ukuhlubula 5.4 cm ubude ngaphansi ukucatshangelwa kusho isetshenziswa isikhumba endaweni oyifunayo futhi ukuzihlikihla ezithambile massaging ukunyakaza kuze ukumuncwa yayo egcwele.
Kufanele kuqashelwe ukuthi ezinkudlwana endaweni endaweni ethintekile, kulapho izidakamizwa ingena yokumelapha. Ngakho strip pyatisantimetrovym nomuthi "Artrokol" kulingana 100 g ketoprfena.
Ngemva okugcoba isetshenziswa, kufanele ngokushesha geza izandla.
ijeli Okubukwe ovunyelwe ukusebenzisa ngokuhlanganyela nezinye ukuthaka imithi oqukethe ketoprofen (isib ngokuhlanganyela amaphilisi, amaphilisi, suppositories rectal).
Umthamo esiphezulu ejenti 200 mg ngosuku. Lona inani izidakamizwa akuxhomekile ngendlela imithi.
Ubude Yiqiniso zokwelapha kufanele sizimisele njalo ngamunye udokotela ukuba khona. Nokho, kufanele kuphawulwe ukuthi liniment ukusetshenziswa izinsuku ezingaphezu kwezingu-10 ilandelana akuvunyelwe.
Imiphumela engemihle
Imiphi imiphumela emibi ongaba kubangele izidakamizwa "Artrokol" (gel)? Ukufundiswa elikushoyo miphumela elandelayo engakhi imvelo:
- bronchospasm, angioedema;
- ukuhlaselwa isifuba somoya, ukusabela anaphylactic ehlanganisa ukushaqeka;
- ububomvu, ukulunywa, ukuqubuka, evutha nokuvuvukala kwesikhumba;
- bullous phlyctenular eczema nonekhono esakaza kwezinye izindawo futhi ukuthola generalized;
- photosensitivity, bullous noma xhumana dermatitis;
- isicanucanu, Stevens-Johnson syndrome, ukuhlanza;
- ukopha, izilonda esiswini, uhudo, isilungulela, ukuqunjelwa;
- Ukuphazamiseka umsebenzi izinso, exacerbation of kwezinso ukwehluleka imvelo okungamahlalakhona, nephritis interstitial kanye nokwehluleka kwezinso.
Kufanele kuphawulwe ukuthi uma usebenzisa ijeli "Artrokol" kungababangela ezinye ohlangothini ukusabela futhi lomgudu wokugaya ukudla bese uhlelo urinary. Amandla miphumela incike inani izidakamizwa futhi permeation ikhono isithako yayo iyasebenza, endaweni iphathwa usayizi, izinga kanye nesikhathi isimo zokwelapha kwesikhumba.
Asinakusho ukuthi asebekhulile sibuthakathaka kakhulu ukuba imiphumela emibi ama-NSAID ekwelapheni.
Phakathi nokukhulelwa kanye lactation
Ngingakusebenzisa kanjani lokhu izidakamizwa "Artrokol" (gel) ngenkathi bekhulelwe nangenkathi bencelisa? Ngokuhamba ucwaningo amagundane, kwatholakala ukuthi izimali akakubangeli umphumela teratogenic futhi embryotoxic e izilwane ezisencane. Nokho, kufanele kuphawulwe ukuthi umphumela encane embryotoxic okuye kwaqashelwa ukulinga onogwaja.
Njengoba ukuphepha ketoprofen kwabesifazane abakhulelwe engakaze kusekelwa iyiphi imfundo, ochwepheshe musa batusa ukusebenzisa leli thuluzi ukuze omama abakhulelwe.
Futhi kufanele kuphawulwe ukuthi ketoprofen nezinye inhibitor ka prostaglandin zamagama kungaba avuse ubuthi kwezinso, yamaphaphu futhi izinhlelo inhliziyo umbungu.
Imikhiqizo ukubola izimali zitholakala ngobisi lwebele. Ngenxa yalesi sizathu, ijeli "Artrokol" akufanele zaphathwa abesifazane asebekhulile.
ulwazi oluthile
Ukulungiselela "Artrokol" (gel), okuyinto analogs tibalwe lapha ngentasi, ke kungavunyelwe ukusebenzisa ezindaweni isikhumba nezinguquko sokugembula ezifana induna noma eczema. Kuyefana nasendleleni endaweni onegciwane noma izilonda ezivulekile.
Kufanele ugweme contact izidakamizwa kanye nolwelwesi lwamafinyila. Ngemuva kokusebenzisa izidakamizwa kufanele ageze izandla zawo.
Leli thuluzi asifanele ukusetshenziswa ne kusaladi occlusive.
Phakathi ukwelashwa "Artrokolom" futhi amasonto amabili emva kokwelashwa, kuyinto efiselekayo ukuze zigweme ukuthintana isikhumba elangeni.
"Artrokol" (gel): ukubuyekezwa kanye amalungiselelo efanayo
Ngu analogue yalesi izidakamizwa ahlanganisa izidakamizwa ezifana "Karmolis-ijeli", "Indomethacin", "diclofenac", "Remisid", "Vipratoks", "Denebola", "Injongo T", "chondro-amandla", "ibuprofen" "Ketonal" nabanye.
Okushiwo ngabantu mayelana abasebenzisa izidakamizwa? Babika ukuthi ijeli "Artrokol" limelela umenzeli ngempumelelo eqeda ukuvuvukala. It ephatha kahle labo izimo zokucabanga okubangelwa isifo efana myalgia, izifo kohlelo locomotor, Izifo ukuvuvukala ka imithambo ukuvuvukala ukucindezeleka kwangemva kwenhlekelele.
I yokuntula lokhu imithi lokusebenza olungaphandle zihlanganisa sebuningini ohlangothini-imiphumela okuyinto azibonakali ngemva gel ukusetshenziswa. Ngokuvamile, iziguli ebonwe ububomvu, ukulunywa, isifuba esivuthayo nokuvuvukala kwesikhumba, kanye nesicanucanu, eczema, izilonda esiswini, isifo sohudo kanye isilungulela. Enye kusimo zomuthi kubhekwe ukuthi asikwazi ebekiwe kwabesifazane abakhulelwe, kanye ukusetshenziswa phakathi lactation.
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