Impilo, Amalungiselelo
Umuthi 'Tizanil ": yokusetshenziswa, analogs kanye nokubuyekeza
"Tizanil" - a relaxant imisipha, ukuhlinzeka isenzo emaphakathi. Ukuze wehlise ithoni imisipha yohlaka wayevame izidakamizwa "Tizanil" izinkomba ukusetshenziswa okukuvumela, uma kunesidingo, ukususa kwemisipha izinhlungu zibe eziwumphumela ukuthuthukiswa isifo esithinta izinzwa, esiwohlozayo disc isifo, ukuhlinzwa noma ukulimala. Ngaphandle esebenzayo isithako tizanidine, le nomuthi yakhiwa izingxenye ezengeziwe. umphumela Asizayo kungenxa yokuba khona Silicon dioxide, stearic acid, microcrystalline cellulose futhi monohydrate-lactose.
isinyathelo kwemithi "Tizanila"
receptor Alpha2-adrenergic ocushiwe futhi ngemva kokwamukela "Tizanil" lisho ukuthini. Ukwakheka ekwakhiweni ungakwazi ukubhekana ngempumelelo nge amajaqamba babazi wabonakaliswa futhi zibe ifomu okungamahlalakhona, osiqalo sakhe sisukela palsy noma umgogodla. Lokhu ejenti kusiza ukunciphisa imisipha ukumelana ngesikhathi ukunyakaza yekwentiwa kanye ukwandisa ngokungenasizathu Kufinyeta kwemisipha.
Absorption zomuthi kwenzeka ngokushesha. "Tizanil" yokusetshenziswa kunjengesipho ithuluzi amuncwa umzimba cishe ngokuphelele inani eliphezulu atholakala igazi imizuzu 60 ngemva kokufaka ipheshana wokugaya ukudla.
Umzimba kwenzeka isibindi, bioavailability oluhambisana 34% sesibopho ukuthobisa plasma amaprotheni - 30%. Engxenyeni-ukuphila ithatha isilinganiso samahora amathathu. Umuthi is excreted kusuka emzimbeni njengoba metabolites ikakhulukazi izinso, isabelo saso encane sisuswa njengoba yayinjalo.
ubufakazi
Okukushoyo "Tizanil" izinkomba ukusetshenziswa zimi kanje:
- emgogodleni isifo kwemisipha izinhlungu zibe, okuyinto ahambisana ubuhlungu;
- buhlungu imisipha zibe ngemuva kokuhlinzwa;
- lwamathambo imisipha spasticity ngenxa izifo zezinzwa.
Izimo ethola "Tizanila"
Imithi contraindicated nge hypersensitivity kuya izingxenye zalo, iziyaluyalu isibindi kanye nezinso, kokuba libizwa. "Tizanil" imfundo ayikuvumeli ukusebenzisa ngesikhathi sokukhulelwa wengane kanye webele ukusuthisa kuye. Contraindication kuyinto ekwelapheni "fluvoxamine". Ubudala esingaphansi iminyaka engu-18, futhi sisebenza Izimo.
Ngo esingamahlalakhona kwezinso, ukulaya ivumela ukusetshenziswa kwezidakamizwa, kodwa ngokucophelela okukhulu. Kuyefana nasendleleni ukusetshenziswa ahlangene "Tizanila" nge CYP1A2 inhibitor nokwelashwa kwasebekhulile.
Isicelo nomuthi Isikali
Umuthi esithathwayo ngomlomo. Uma injongo ukusetshenziswa kwezidakamizwa ukushabalalisa buhlungu imisipha zibe, kutuswa ukusebenzisa umthamo ezisukela 2 kuya ku-4 mg. Umthamo watusa amanxusa kumele kuthathwe kathathu ngosuku. Uma kwenzeka kuba nzima, it ovunyelwe ungeze zinsiza obengeziwe 2-4 mg nomuthi "Tizanil". Izibhebhe ngokuvumelana Umhlahlandlela isicelo ingasetshenziswa kwemisipha lwamathambo spasticity 6mg. Lona umthamo sangemihla, okuyinto lapho besanda kuqala ukwelashwa akufanele kudlulwe. Ekwelapheni izifo ezifana Kwenziwa ezintathu nokushintsha kokudla nokufakwa nsuku zonke. Ukuqaphela isikhawu 3-7 izinsuku ka, umthamo kungenziwa kancane kancane nge-avareji ka-3 mg.
Ukuze umphumela esiphezulu, ngokuletha kuvunyelwe umthamo wansuku zonke ukuze 24 mg. Umthamo elikhulu ngokuvamile 12 mg noma ngaphezulu, kodwa awukwazi ukudlula 36 mg. Ngakho nsuku zonke kufanele kwenziwe 3 noma 4 eyamukelayo kusho "Tizanil". Yokusetshenziswa iqukethe ulwazi nokwelashwa kweziguli esingamahlalakhona kwezinso. Iziguli ezinjalo ekuqaleni ezinqunyiwe izidakamizwa ukusetshenziswa kanye ngosuku umthamo ubuncane elihambisana 2 mg. I Isikali is kancane kancane washintsha ukusabela isiguli. Uma ufuna ukwandisa umthamo, okwandisa komthamo wokuqala kakhulu, bese ukushintsha inani isibalo.
side effects
ukwelashwa isikhathi eside ngezinye izikhathi ephelezelwa ukusabela engathandeki umzimba. Kulokhu, bangakwazi ukuhlakulela kakhudlwana futhi avele evelele. Lokhu kusebenza futhi yokwamukela ngemithamo enkulu "Tizanil" izidakamizwa. Yokusetshenziswa Ngokusho miphumela emibi, njengoba ukungasebenzi pheshana emathunjini, iphele we ulwelwesi lwamafinyila emlonyeni, ukwehla abangelutho wegazi, ukutubeka komzimba, ukozela, isiyezi kanye nezinye izigigaba ezingezinhle.
Ukuvela amathuba okuba nemiphumela engemihle kuba isizathu ukwelashwa udokotela, okuyinto noma ukunciphisa umthamo noma ukukhansela izidakamizwa, esikhundleni sako ulethe ngezinye izindlela. Ngo amaphilisi ukwelashwa "Tizanil" yokusetshenziswa kufanele waphawula ukuthi ingozi nemiphumela engathandeki yalawo maphilisi lincishisiwe.
izidakamizwa ekuhlanganyeleni
Ukuxhumana kwemithi ezahlukene - lena ukwaziswa okubalulekile kakhulu, okumele kubhekwe ngaphambi kokwelashwa ukuze unciphise amathuba okuba nemiphumela engemihle, okuhlukile ukulimaza umzimba futhi kuncishiswe ingozi ukusebenza yokwelapha.
Kuyaziwa ukuthi lesi sidakamizwa "Tizanil" kuhlangene 'Fluvoxamine ", kuholela Ukuwohloka impilo. Lapho-ke concomitantly nezidakamizwa antihypertensive ingaqala bradycardia futhi hypotension.
Uma bobabili Ethanol noma sedatives kanye amaphilisi "Tizanil" imfundo kubonisa ukwanda ukupholisa, okuyinto Ilungiselelwe "Tizanilom". Nge inhlanganisela yakhe izinto zokuvimbela inzalo temlomo singanciphisa imvume nengxenye.
Izidakamizwa ekusebenzisaneni Ungashintsha kusebenta ukwelashwa. Ngekusetjentiswa kanyekanye izidakamizwa eziningana, bangase ukuthuthukisa umphumela nomunye noma sicindezeleke. Konke lokhu igcwele ukubukeka ukusabela ezingezinhle, ukweqisa izidakamizwa, zintula umphumela kunesidingo.
Izixwayiso
Ngaphambi kokuqala imishanguzo "Tizanil" Izinkomba kanye contraindications kumele uzifunde ngokucophelela.
Kuthiwa okuvela izinguquko olunzulu nezinso isibindi. Kodwa nge ukwelashwa okusekelwe ngokuthatha izidakamizwa umthamo 12 mg noma ngaphansi, amacala anjalo kwakungamelwe ivelakancane.
Kutuswa ukuthi ngezikhathi ezithile ukuthatha umsebenzi ukuhlolwa isibindi. Phakathi nezinyanga zokuqala ezingaba zine - ngenyanga esisodwa. Ezimweni lapho AST no-ALT amazinga angaphezu amagugu evamile kakhulu uyeqe, kudinga ukuqedwa zomuthi.
Ezinye iziguli abathatha "Tizanil" (kuhlanganise analogs) zingavela ukozela. Nakuba kulesi sifundazwe, awukwazi benze umsebenzi odinga bagxila futhi ukusabela okusheshayo.
Ngenxa usongo ukuwohloka isiguli izidakamizwa is okungazange kukhanselwe ngokuzumayo, it is yalahlwa kancane kancane umthamo ukunciphisa.
Analogs "Tizanila"
Letibekiwe imiyalelo sikhungo "Tizanil" Ukufundwa akusho ngaso sonke isikhathi ukuba usebenzise original ngenxa ezinye Izimo. Izidakamizwa eqolo eyakhe "tizanidine-Teva" futhi "Tizalud". Le mithi futhi relaxants, etholakala ifomu tablet babe isithako efanayo esebenzayo.
Manufactured nezinye analogs. Ngokwesibonelo, zokwelapha kungase kube into "Mydocalm", "Teva-Tizanilom" Surdaludom MR "," Surdaludom ".
Izibuyekezo
Uphenyo "Tizanile" awafani, isb. Ukuze. Umuthi kungathinta iziguli ehlukile. Kodwa izikhathi eziningi zingabantu omuhle. Lesi sakhiwo baqala ukunyathelisa isikhathi eside, isendalini isikhathi eside, abantu abaningi kangaka beye bakwazi ukuqinisekisa ukusebenza yayo. Kukhona Izibuyekezo ezingezinhle kwesokunxele isizathu nemiphumela engemihle ngenxa ukungabekezeleli izingxenye noma ukusetshenziswa ngemithamo ephakeme Kunconywa for ekwelapheni "Tizanil" izidakamizwa. Izibuyekezo ezinhle kwesokunxele abantu bayajabula umphumela, enqubeni ukwelashwa athobele Isikali ebekwe udokotela, futhi cishe abazange bakuqaphele ngasiphi abantu basabele ngendlela embi.
umuthi ngokuvamile asetshenziselwa ukwelapha esiwohlozayo disc isifo. Ngenxa izimpawu zaso isenzo ezihambisana nalesi sifo zinyamalale ngokushesha. Dlulisa ikhanda futhi ubuhlungu emuva, kuthuthukisa impilo jikelele. Ngezinye izikhathi kukhona kabi imithi emzimbeni okungatheni ezifana ukozela, kome le mucosa ngomlomo, kodwa ukulungiswa efanele umthamo noma kuhoxiswe lokho izidakamizwa ayanyamalala. Ezinye iziguli nge acute egeleza osteochondrosis, avuse radicular syndrome, okungukuthi 'Tizanil "wabuya ukuhamba evamile, kanti eminye imithi akangayiletha imiphumela oyifunayo.
Umuthi akuyona kususa okubi okusezingeni eliphezulu imisipha ithoni, egcwele phetho unhlangothi. "Tizanil" kuthathwe kuphela kadokotela ebukhoneni izinkomba ezifanele. Uma impatho liyadingeka umuntu osekhulile noma isiguli isibindi onesifo, kungcono hhayi ukuba engozini impilo bese ukhetha imisipha relaxant ezahlukene, okuyinto futhi ubhekana kahle imisebenzi.
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