ImpiloAmalungiselelo

"Truksal": ukubuyekezwa odokotela. "Truksal": yokusetshenziswa, side effects

Bambalwa abantu bazi, kodwa sengqondo, neurosis nokucindezeleka amenable ekukhetheni izindlela zokwelapha. Okubaluleke kakhulu, isikhathi ukuze ujike i abanolwazi kanye ngokuqinile zonke izincomo zayo.

Ngokuvamile, ngaphansi kwezimo ezinjalo e antipsychotics iziguli ebekiwe noma kangaka okuthiwa neuroleptics. Bona kakhulu ukunciphisa izimpawu kuphazamiseka ingqondo, kubuyisele nesineke isizathu okumsulwa futhi ukucabanga ngendlela esile.

The njalo kunazo ebekiwe lapho izifo eziphawulwe ngenhla okunzima nomuthi ezifana "Truksal". Qaphela, impendulo, contraindications ukusabela ezingezinhle zomuthi uzobe kuchaziwe ngezansi.

Ubujamo, incazelo, emabhokisini kanye nokusungulwa

I nomuthi "Truksal" (Physicians izilinganiso kuyothiwa elichazwa kamuva esihlokweni) ikhiqizwa njengendlela amaphilisi obunsundu round namafomu biconvex, ifilimu-camera.

ekwakhiweni Okubukwe iqukethe isithako ezifana chlorprothixene hydrochloride. Lihlanganisa izingxenye ezengeziwe njengoba corn isitashi, copovidone, monohydrate lactose, glycerol, microcrystalline cellulose, talc, sodium croscarmellose kanye magnesium stearate.

Ngokuphathelene ifilimu enamathela, liphethe hypromellose, Macrogol 400, obomvu yensimbi oxide, ensimbi amnyama oxide ne-titanium dioxide.

Ngo iphakheji wanikela ukudayiswa "Truksal" ithebhulethi? Izibuyekezo Umthengi wazise ukuthi emashalofini Pharmacy izidakamizwa ingatholakala amakhadibhodi amaphakethe, aqukethe nezipakupaku.

umphumela we izidakamizwa

Uyini izidakamizwa "Truksal"? Izibuyekezo ochwepheshe ukubika ukuthi lena izidakamizwa ngempumelelo kakhulu. Kuyinto izidakamizwa antipsychotic (isb neuroleptic) kanye esuselwe thioxanthene.

Lo muthi unamandla ukunikeza antidepressant ngokulinganisela, sine nemiphumela antipsychotic.

Impahla yokugcina izidakamizwa ngenxa yekhono layo ukuze uvimbele Dopamine receptor. Nge isenzo esinjalo futhi ahlobene nomuthi analgesic nemiphumela antiemetic.

Ngokusho imfundo, "izilinganiso Truksal 'zazo axutshwa, nje kuphela abazokwazi ivimbela i-alpha-1 adrenoceptors futhi serotonin 5-HT2-receptor, kodwa histamine H1-receptor. Lokhu kubangela antihistamine, antihypertensive futhi adrenoceptor Ukuvinjwa yayo senzo.

I kinetics kwezidakamizwa

Kungakhathaliseki imithi ugxile "Truksal"? Izibuyekezo Umthengi ngeke uyithole impendulo yalo mbuzo. Ngemuva ke kuyomelwe emiyalelweni noma abanolwazi. Ngokusho kwabo, ngemuva kokuthatha izidakamizwa ngaphakathi Chlorprothixenum angabacwasi ngokushesha ugxile kusukela pheshana emathunjini.

Umkhawulo igazi lokuhlushwa izidakamizwa esebenzayo siyenzeka emva kwemizuzu 120. I bioavailability zomuthi kuyinto 12%.

Kufanele futhi wazi ukuthi Chlorprothixenum lingena sasivumela kalula ngokusebenzisa isithiyo esinomhlapho futhi ngesilinganiso esincane excreted ne ubisi.

Isigamu-ukuphila ithuluzi amahora 16. I metabolites okuholela unomsebenzi neuroleptic. Basuke okukhonjiswe indle kanye nomchamo.

ubufakazi

Kungaphansi kwaziphi izimo ziboniswa iphilisi "Truksal"? Uphenyo odokotela bathi ukuphumelela kwalesi izidakamizwa evelele kakhulu lokuchezuka ezilandelayo:

  • ukuhoxiswa syndrome lapho yizidakamizwa nokuluthwa utshwala;
  • kwengqondo kuhlanganise uthi ukwenama, ukusangana, ukuyaluza, ukuyaluza nokukhathazeka;
  • ezibangela ukuziphatha okuyinqaba ezinganeni;
  • hyperactivity, ukuyaluza, ukucasuka, ukudideka kwasebekhulile;
  • ukuqwasha;
  • uthi futhi bacindezeleke, iziyaluyalu futhi neurosis zengqondo;
  • ubuhlungu syndrome (lihambisana analgesics).

Izimo

Ngokusho imiyalelo, ethola neuroleptic "Truksal" is contraindicated ku:

  • pheochromocytoma;
  • nokuquleka ngenxa yokuphuza kakhulu ;
  • CNS ukucindezeleka Lokudabuka ehlukahlukene (kuhlanganise utshwala, analgesics opioid futhi barbiturates);
  • yezifo igazi;
  • ibele;
  • nciphisa semithambo;
  • ukhulelwe;
  • hypersensitivity kuya izithako zako.

Tablets "Truksal": yokusetshenziswa

ochwepheshe lezivakashi bathi lokhu imithi kumele isetshenziswe kuphela ngenjongo udokotela abanolwazi. Uma kungenjalo, kungenzeka neqhaza ekuthuthukiseni engalawuliwe reception sebuningini ukusabela kwalo.

I umthamo we-ejenti incike uhlobo lwesifo.

Ngo kwengqondo kanye bayasangana uthi ukwenama ekuqaleni ukwelashwa le nomuthi iqondiswa ngezilinganiso ka 50-100 mg ngosuku. Ngaphezu kwalokho, inani ukulungiswa luyanda ku-300 mg ngelanga (ngezinye izikhathi afinyelela ku-1200 mg). Lokhu Isikali sehlukaniswe 3 ngemithamo.

Ekwelapheni kwezimpawu zokuqaleka nge yizidakamizwa nokuluthwa utshwala umthamo wansuku zonke imithi kufanele kube mg 500 ngezinyathelo ezintathu. Inkambo yokwelashwa - ngesonto elilodwa.

Asebekhulile ebukhoneni ukucasuka, ukuyaluza, ukudideka noma hyperactivity ukwazi nomuthi iqondiswa i inani 15-90 mg ngelanga (imithamo emithathu).

Izingane ukulungisa ukushayisana ukuziphatha izidakamizwa kunikezwa ngesilinganiso umthamo 0.5-2 mg ngayinye kg esisindo.

Uma ayimigodi, elihlanganiswa ukucindezeleka nokukhathazeka, amaphilisi "Truksal" ingasetshenziswa njengendlela monotherapy, njengenhlangano ezama ukubuyisa adjunct ukuze ukwelashwa nge antidepressant.

Lapho iziyaluyalu zengqondo neurosis, neziyaluyalu bacindezeleke ezihilela ukukhathazeka, nomuthi Kunconywa ukusebenzisa umthamo 90 mg ngelanga (imithamo emithathu).

Ngenxa yokuthi lokhu izidakamizwa akakubangeli ukuluthwa noma sezidakamizwa, ingasetshenziswa isikhathi eside.

Lapho ukuqwasha namaphilisi ukuba 20-30 mg kusihlwa futhi ihora elilodwa ngaphambi sokulala.

Izidakamizwa "Truksal": ukubuyekezwa, side effects

Njengazo zonke antipsychotics, izidakamizwa kubhekwe ngokuvamile kubangela imiphumela eminingi engemihle njengezindlela :

  • somnolence, izimpawu extrapyramidal, isiyezi, yokuhlala thuthuva;
  • tachycardia, hypotension orthostatic ;
  • nomlomo owomile, jaundice cholestatic, ukuqunjelwa;
  • dysmenorrhea, buthakathaka potency, galactorrhea;
  • kwesisindo anda ukujuluka, isifiso sokudla kakhulu;
  • anaemia Hemolytic, leukopenia, lezivakashi ingozi;
  • ukuqubuka.

Izibuyekezo mayelana leli thuluzi zingaphezu omuhle. Kaningi umama ngaye ukhuluma izingane ezibangela ukuziphatha okuyinqaba. Bathi umuthi ayizwakali.

Ngokuqondene odokotela, izimpendulo zabo awavamile. Waleyo, kuphephile ukuphetha ngokuthi izidakamizwa esimweni ngasinye sikhombisa umphumela ohlukile.

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