ImpiloAmalungiselelo

Medicine 'carvedilol'. Yokusetshenziswa

Medicine "Carvedilol", ngokuvumelana iziguli, has a action mnene futhi ngempumelelo. Umuthi uyilungu leqembu ejenti antihypertensive.

Kusho "Carvedilol". incazelo

Mshini kwezidakamizwa ukuchayeka esekelwe nokuvinjelwa beta 2, beta 1, i-alpha 1-adrenoceptors. Ngazo izidakamizwa "Carvedilol" yokusetshenziswa libhekisela ikhono layo ngokulinganisela ukwehlisa conductivity, nobuningi namandla ukusikwa inhliziyo, ngaphandle ingqondo a bradycardia abukhali. Nokuvinjelwa kwe-alpha-1 adrenoceptors kwabangela ukwanda kubangela izitsha neuropathy. Lapho ukuvinjelwa beta ithoni 2-adrenergic kwandisa kancane kwezinye izitsha microvasculature, ukucinana kwemigudu yokuphefumula, kanye ithoni bese peristalsis emathunjini.

Medicine "Carvedilol" Umhlahlandlela uncoma nomfutho wegazi ophezulu.

Yabela izidakamizwa ngaphakathi. Ezinsukwini zokuqala okwelashwa, umthamo 12.5 angu esisodwa. Ngemva nenani lomuthi luyanda kabili (25 mg). Futhi thatha kanye ngosuku. Ngokusho isincomo udokotela, uma kunesidingo, umthamo we izidakamizwa "Carvedilol" imfundo on isicelo uvunyelwe ukwandisa. Ningaphathi usuku angu ezingaphezu kwamashumi amahlanu. Ukwanda Isikali kumele akenzanga okungaphezu kokukodwa ezinsukwini eziyishumi nane. Ukuze ezigulini esezikhulile nekusebenta kungabonakala nasemkhakheni uma nithatha 12.5 angu.

ukubonakaliswa Esibi zomuthi "Carvedilol" imfundo on isicelo siphathelene iziqephu ngokweqile ingcindezi ukunciphisa. La machashazi abizwa kuphawuliwe ekuqaleni yokwelapha ( "lokuqala umthamo syndrome") futhi ukwanda okwalandela e nenani lomuthi wathola. Njengomthetho, lezi uthi ziyasuswa ngokuzimela ngaphandle kokudinga Isikali izinguquko.

Ukusetshenziswa okwalandela zomuthi "Carvedilol" kungaba liyochukuluza nokuqinisa motility emathunjini bese ithoni, bradycardia, ubuhlungu bekhanda, ukukhathala, ubuthakathaka. Libuye angina kungenzeka, iziyaluyalu kwegazi neuropathy, lomkhuba ka claudication ngakanye. ukubonakaliswa Esibi zomuthi "Carvedilol" yokusetshenziswa futhi lidlulisela okubi kakhulu wefayela psoriasis langaphambilini, urticaria, ukusabela ezihlobene ekuthuthukiseni ulele planus, exanthema nomzimba.

Ezimweni ezingavamile, izidakamizwa kungabangela leukopenia, ekhaleni stuffy, thrombocytopenia, kukhuphuke ukumelwa inhliziyo, paresthesia (ndikindiki), ukucindezeleka, unenkinga.

Medicine "Carvedilol" contraindicated e atrioventricular block wesibili noma degree lwesithathu, ukushaqeka, decompensated ukuhluleka kwenhliziyo, isifuba somoya, yokwehluleka kwesibindi, izifo zamaphaphu nzima nge BOS syndrome, hypersensitivity emuthini. Hhayi esimisiwe ejenti lactation ngesikhathi sokukhulelwa.

Izixwayiso

Medicine "Carvedilol" okunqunyiwe ngokuqapha in iziguli senhliziyo futhi yenhliziyo Umthambo isifo. Ephambi kwezinduna inhliziyo ukwehluleka ngaphambi ukusebenzisa izidakamizwa kuyadingeka ukuze ukuqhuba ukwelashwa okufanele ukuze aqede kuwukubonakaliswa decompensation. In iziguli yenhliziyo Umthambo isifo kanti ukuthatha izidakamizwa, "Carvedilol" kungehlisa izinga esivimba amanzi nomoya-mpilo funa. Kule ndaba, ukuqedwa zomuthi wenziwa kancane, ukugwema ukuthuthukiswa zokuhlasela angina.

Phakathi ukwelashwa belulekwa ukugwema utshwala.

Ekuqaleni yokwelapha kanye lapho okwandisa umthamo kufanele uyeke ekufezeni imisebenzi engase ibe ingozi, kuhlanganise nokuphathwa kwezokuthutha.

Ngaphambi kokusebenzisa izidakamizwa "Carvedilol" kubalulekile ukuba sihlole isifinyezo, xhumana nodokotela.

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