EzempiloAmalungiselelo

Iyini iPiracetam esetshenziselwa? Imiyalo yokusetshenziswa "iPiracetam"

Kungani iPiracetam inqunyelwe iziguli? Impendulo yalo mbuzo uzofunda kulokhu kulesi sihloko. Siphinde sikunike ulwazi mayelana nokuthi ungathatha kanjani lo muthi, ngukuphi uhlobo olukhishwayo, kungakhathaliseki ukuthi unemiphumela emibi kanye nokuphikisana, kungakhathaliseki ukuthi kungasetshenziswa ngesikhathi sokukhulelwa futhi ngesikhathi sokukhulelwa.

Amafomu okulungiselela, ukupakisha nokubunjwa

Ngaphambi kokuba usitshele ukuthi yikuphi "iPiracetam" enqunywe odokotela, kufanele usitshele ukuthi iyiphi into engathengwa kuma-pharmacy.

Namuhla kunezinhlobo eziningana zalesi sidakamizwa. Ake siwahlole ngokuningiliziwe.

  • Amaphilisi. Leli fomu lezidakamizwa liqukethe u-0.4 g we-piracetam futhi lidayiswa ngamaphakheji ekhadibhodi wezingcezu ezingu-60.
  • Isixazululo se-20%. Leli fomu lidayiswa ngama-ampoules ka-5 ml, okubekwe wona, afakwa emaphakheji ekhadibhodi wezingcezu ezingu-10.
  • Amathebulethi. Isidakamizwa siboshwe ngengubo ephuzi futhi iqukethe u-0.2 g wezinto ezisebenzayo. Ungathenga amaphilisi emaphaketheni wekhadibhodi angu-120 noma izingcezu ezingu-60.
  • I-granules yezingane. Isidakamizwa sinombala okhanyayo obomvu (tshela i-brownish sediment), itholakala ezigodini zemibukiso ngo-56 g.

Kumele kuqashelwe ukuthi ifomu ngalinye lezidakamizwa linempahla yalo eyisizayo.

Pharmacodynamics of the izidakamizwa

Kungani "i-Piracetam" ingabelwa umuntu? Kuyinto imithi ye-nootropic engaba nomthelela omuhle ekusakazeni kwegazi kobuchopho kanye nezinqubo zayo zokusebenzisa umzimba.

Le mithi ithuthukisa izinqubo ze-metabolic futhi yandisa ukusetshenziswa kwe-glucose. Ibuye ivimbele ukuhlanganiswa kwamaplatelets acushiwe.

Ukwamukela "i-Piracetam" kunomphumela wokuzivikela ekulimazeni komqondo, okubangelwa ukwethuka kagesi, ukudakwa noma i-hypoxia. Ngaphezu kwalokho, lesi sidakamizwa sithuthukisa umsebenzi wokuhlanganiswa kobuchopho, ngaphandle kokusebenzisa umqondo wokuguqula umzimba nokudambisa.

Izakhiwo zomuthi

Yiziphi izindawo zomuthi "iPiracetam"? Iyini injongo yalolu remedy? Lesi sidakamizwa sikwazi ukuvuselela izinqubo zokusebenzisana ohlelweni lwezinzwa eziphakathi, nokuthuthukisa isimo sengqondo nokukhumbula inziguli ezimbili kanye nabantu abanempilo.

Kungani "i-Piracetam" ingabelwa izingane? Leli thuluzi liyakwazi ukwandisa umsebenzi wezingqondo, ukuthuthukisa ukusebenza kwengqondo, ukwenza ngcono izinqubo zokufunda, ukuthuthukisa ukuqhutshwa (synaptic) ku-cortex ye-cerebral kanye nokuxhumana phakathi kwama-hemispheres (kwesobunxele nangakwesokudla). Futhi, umuthi ubuyisela futhi uzinzisa inkulumo ephazamisayo, inkumbulo nokuqonda.

Isimiso sokusebenza komkhiqizo wokwelapha

Isidakamizwa "iPiracetam" sisebenza kanjani? Kungani abantu bakhe abasebasha kanye nabantu asebekhulile basebenzisa?

Lesi sidakamizwa simisa isilinganiso se-ATP ne-ADP, futhi siphinde senze i-phospholipase A, ivuselele ukushintshaniswa kwama-neurotransmitters futhi ikhuthaze ukugqugquzelwa kwezinqubo zeplastiki nezenzakalelo ezinamathisini omzimba.

Ngabe yikuphi "i-Piracetam" (imijovo, i-powder, i-capsules namathebulethi) angahle anqunywe iziguli? Lesi sidakamizwa sikwazi ukuvimbela ama-platelet aggregation, ukuthuthukisa ukucwiliswa kwemithi kanye nokwandisa ukuhamba kwamaseli abomvu obomvu ngemikhumbi encane.

Kufanele kuphawulwe ukuthi le nsizakalo ikwandisa ukujikeleza kwegazi kwesifunda ezindaweni eziyi-ischemic zobuchopho, ithuthukisa umsebenzi we-alpha ne-beta, kodwa inciphisa umsebenzi we-delta.

Imithi iyanciphisa i-vestibular nystagmus. Nge-hypoxia, ukuhlukumezeka nokudakwa, kusebenza umphumela we-neuroprotective.

Ngokuqondene nezindawo ezingenayo i-antihypoxic le mithi iphumelela kakhulu ekwelapheni okuyinkimbinkimbi ye-infarction ye-myocardial.

Pharmacokinetics yomuthi

Isidakamizwa "Piracetam" sithatha isikhathi esingakanani (siyini injongo yalolu remedy, sizoxoxa kamuva)? Ngemuva kokungenisa, isidakamizwa sisheshe siphume ngokuphelele. I-bioavailability yayo ayikhulu ngamaphesenti.

Ukuphathwa komlomo ngomuthi ngenani lika-2 g unikeza ukuhlushwa okuphezulu ku-plasma emva kwemizuzu engamashumi amathathu. Isidakamizwa asibophezeli kuma-protein, singena kuzo zonke izitho kanye nezicubu, kufaka phakathi nomgoqo ophansi.

Isidakamizwa cishe asihlanganisi kahle, kodwa sikhetha ngokuqoqa ezindaweni ezihamba phambili ze-parietal, ze-occipital nezangaphambili zobuchopho, kanye ne-cerebellum ne-basal ganglia.

Ingxenye yokuphila yalesi remedy amahora amahlanu. Cishe i-95% yalesi sidakamizwa sidonswe emcinini ongashintshi (ngemuva kwamahora angamashumi amathathu). Kubantu abanezinkinga zezinso lesi sikhathi sesikhathi sanda.

Iyini i-Piracetam? Izinkomba zokusetshenziswa

I-agent ye-nootropic ecatshangelwe inezinyathelo eziningi. Ngokomyalelo, izinkomba zokusetshenziswa kwazo zilandelayo:

  • Isifo so-Ischemic, kanye nayo yonke imiphumela yaso;
  • Ukungaqiniseki komzimba ongapheli (isib. Ukushona kwe-atherosclerosis, isifo esiwumfutho wegazi noma i-parkinsonism yama-vascular), ehambisana nezinhloko, isizungu, inkumbulo, inkulumo nokukhathazeka kokukhathazeka;

  • I-Dementia (kuhlanganise nesifo se-Alzheimer);
  • Aphasia;
  • Ukuvuthwa kwe-viral neuroinfection (acute);
  • Izifo zesimiso sezinzwa, ezihambisana nokunciphisa emisebenzini yengqondo kanye neyemnestic, izinga lokuvuka, kanye nokwephulwa komkhakha wemizwelo nokuzimelela, ukuziphatha;
  • Ukuxila (kuhlanganise ngesikhathi sokuphumula, i-subcomatose ne- coma) ;
  • Isizungu;
  • Ukuphazamiseka kwengqondo;
  • Isimo esibucayi nesinandaba;
  • I-myoclonus ye-cortical;
  • I-craneocerebral trauma;
  • Isifo sokuphuza (njenge-adjuvant);
  • I-nystagmus vestibular;
  • Izinqubo ze-Atrophic and senile.

Kuphi ukuphambuka kusalokhu kunqunywe umuthi "iPiracetam"? Kungani baphuza lesi sidakamizwa bese benza imijovo? Ngaphezu kwalokhu okungenhla, le mithi inezinkomba ezifana nalezi:

  • Izinkinga ze-neurological, somatovegetative, ze-psychiatric ezavela emva kokwelashwa ngezidakamizwa ze-psychotropic kanye nama-antipsychotics;
  • Ukudakwa ngokweqile nge-amphetamine, i-ethanol, i-barbiturates noma i-morphine;
  • Izimo ezicindezelayo, ukumelana nokwelashwa ngezidakamizwa zokucindezeleka;
  • Ukucindezeleka kwe-Neurotic ngezingqinamba ze-asthenic ne-senesto-hypochondriacal, kanye ne-adynamics nezimo ze-ideomotor inhibition;
  • Ukuziqhenya, ukulandelelana nokuhleleka okusho ngokudakwa ngokweqile nokulutha izidakamizwa;
  • I-Psycho-organic syndrome enokudakwa ngokweqile (okungapheliyo;
  • I-anemia ye-sickle-cell (ekwelapheni okuyinkimbinkimbi).

Ngoba yiziphi izibhebhe "Piracetam", kanye namaphilisi kanye nodokotela abaphuza njalo batusa ukuba bangenwe iziguli zabo ezincane? Isidakamizwa esinjalo sinqunywe ukukhubazeka kwengqondo encane, ukuphulukiswa kwengqondo, imiphumela yokulimala kwe-CNS yomuntu ngamunye, ikhono lokufunda eliphansi (ne-psycho-organic syndrome), i-oligophrenia, ukuphazamiseka kwenkulumo, ukukhubazeka kwememori nokungaqiniseki kwengqondo.

Ukubamba iqhaza kanye nesikhathi sokubeletha

Ngingathatha yini umuthi "iPiracetam" ngesikhathi sokukhulelwa? Kuyini? Abanye ochwepheshe banikeza umuthi ocatshangelwa abesifazane besimo ngokuvumelana nezinkomba. Kodwa-ke, kufanele kukhunjulwe ukuthi le mithi iwela kalula emkhakheni we-placental, kanye nobisi lwebele. Kulokhu, kukhonjelwa ngesikhathi sokukhwabanisa futhi lapho ubhekene ne-fetus. Uma kungenjalo, kungalimaza impilo yengane.

Ukungafani

Kuziphi izimo ezingenakusebenzisa lesi sidakamizwa "i-Piracetam" (imijovo, amafomu omlomo)? Lesi sidakamizwa asinqunyelwe ukuxoshwa komzimba (kuhlanganise nezidakamizwa ze-pyrrolidone), kanye nesifo sikaHuntington, ukwehluleka okukhulu kwezintuthwane, ukukhulelwa, ukucindezeleka okukhulu, ukushaywa kwesifo esibi kanye nokuncelisa. Futhi, lo muthi awukwazi ukunikezwa izingane ezingaphansi konyaka owodwa.

Izindlela zokusebenzisa

Manje uyazi ukuthi kungani amaphilisi e-Piracetam angabhalwa iziguli. Manje kufanele ukutshele ukuthi ungathatha kanjani lo muthi.

Ekuqaleni kokwelapha, ikhambi le-piracetam lenziwa ngendlela engalinganiselwa ku-10 g. Inani lemithi liyancishiswa futhi lishintshelwa ekulawuleni ngomlomo. Ngaphakathi kwesidakamizwa kuthathwa ngaphambi kokudla kumthamo we-800 mg (ngezilinganiso ezintathu ezihlukanisiwe). Ngemuva kokuthuthukiswa, inani lemithi liyancipha libe ngu-400 mg. Isikhathi sokwelashwa okunjalo ngamaviki ayisithupha kuya kwangu-8.

Kumele kuqashelwe ngokukhethekile ukuthi umthamo wansuku zonke wezidakamizwa "i-Piracetam" ingase ihluke futhi kuxhomeke kuhlobo nobunzima besifo. Ngokuphathelene nobude besikhathi sokwelashwa, kunqunywa udokotela kuphela ngokuhlolwa kwezokwelapha.

Kubantwana ukulungiselela okunjalo ukunikeza okungaphezu kuka 30-50 mg ngosuku. Ngakho ukwelapha kufanele kube yisikhathi eside. Isixazululo sokuphatha ngomlomo sinikezwa ingane izikhathi ezimbili ngosuku (ekuseni nakusihlwa). Kungenziwa wengezwe kumusi wezithelo noma kwezinye iziphuzo.

Ukuphendula okubi

Ingabe ukusebenzisa izidakamizwa "iPiracetam" kungabangela imiphumela engathandeki? Ama-injection, kanye namafomu omlomo wesidakamizwa, akwazi ngempela ukwenza ukuphendula okuhlangene. Okubonakala kakhulu kunazo zonke okulandelayo:

  • I-metabolism: inzuzo yesisindo.
  • Izitho zensiza nesistimu yezinzwa: ukulala, i-hyperkinesia, ukucindezeleka, ukucasuka okukhulu, i-asthenia, ukukhathazeka, ukuhlukumezeka, ukulala kwesifo, ukwanda kobulili, isizungu, ukuthuthumela nokukhanda ikhanda.
  • Ipheshana lokugaya: ukuhlanza, ubuhlungu besisu, isifo sohudo kanye nesicefe.
  • Isikhumba: i-hypersensitivity.
  • Ukusakazwa kwegazi: i- hypotension ye-arterial, i- hypertension, ukungakwazi ukusebenza kwe-coronary (esigabeni sokucindezela).

Overdose

Uma ukudlula ngokweqile komuthi "i-Piracetam" yonke imiphumela emibi ikhuliswa. Njengokwelashwa, kusetshenziselwa isisu esiswini, kanye nokwamukelwa kwamakhemikhali.

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