Impilo, Amalungiselelo
Umuthi 'Relakson ": yokusetshenziswa, incazelo, ukubuyekezwa, analogue
Ngayiphi umthamo ezinqunyiwe zomuthi "Relakson"? Imiyalelo ukusetshenziswa kwezidakamizwa kuzoxoxwa ngezansi. Futhi, uzofunda ukuthi ngabe lokhu imithi analogs babe, ukuthi kubiza malini, lapho kwenzeka aluboniswa, nokunye. D.
Ubujamo, incazelo, ukwakheka kanye nokupakisha
Ukulungiselela "Relakson" ikhiqizwa ngendlela amaphilisi biconvex round ezimhlophe ifilimu-camera. Isithako asebenzayo we umuthi zopiclone. Futhi nomuthi ihlanganisa excipients ezilandelayo: hypromellose, microcrystalline cellulose, i-lactose, amazambane isitashi, colloidal Silicon dioxide, talc, sodium carboxymethyl isitashi, povidone, macrogol, magnesium stearate futhi titanium dioxide.
Ngo iphakheji wanikela ukudayiswa "Relakson" ithebhulethi? Ukufundiswa ukusetshenziswa is ebiyelwe inqwaba amakhadibhodi, okuyinto ezibekwe kanye nentaba yeseli ne izidakamizwa.
izici pharmacodynamic
izidakamizwa "Relakson" Isebenza kanjani? Yokusetshenziswa ibika ukuthi lokhu okuyiluthayo okuqondene tsiklopirrolona iqembu. Ikhipha ke kwehlukile barbiturate futhi benzodiazepine hypnotics. Lesi sidakamizwa kuyinto agonist benzodiazepine yokwamukela. Yokuxoxisana nabo, awusebenzi mbeni la mangqamuzana neuropathy.
izakhiwo zomuthi
Yini property imithi "Relakson"? Izibuyekezo ochwepheshe ukubika ukuthi leli thuluzi uyakwazi ezikhandla, sine okuyiluthayo anticonvulsant omnene, imisipha relaxant futhi tranquilizing imiphumela. Bonke axhunyiwe nge isenzo yokwamukela macromolecular Gaba eziyinkimbinkimbi.
Ngemva amaphilisi kokuthola sithuthukiswe umphumela inhibitory ka Gaba, futhi futhi ukuyiveza ukudluliswa interneuronal ku CNS.
amaphilisi Sleeping "Relakson" kakhulu sifushanise isikhathi sokulala kunciphisa inani awakenings ebusuku ngcono izinga ubuthongo. Futhi, lolu izidakamizwa kwandisa isikhathi sokulala futhi neze kubangela nalawo mathonya postsomnicheskih efana ukozela nobuthakathaka ekuseni.
Habituation ukuze isenzo zomuthi engekho. Ngakho-ke, kungaba zithathwe kuyi imodi batch amasonto 17.
I pharmacokinetics zomuthi
Izidakamizwa "Relakson", intengo oboniswe ngezansi, ugxile ngokushesha futhi kakade emva kwamahora angu-2 siyenzeka egazini. Ukuthola ukudla akuphazamisi ukumuncwa imithi. Ngezinye 45% ke sibopha ukuthi Amaprotheni egazi.
Ngisho nangemva kokuba amasu amaningana ezibhebheni ekuqongeleleni ketshezi asebenzayo futhi metabolites ayifani.
Ingxenye-ukuphila zopiclone futhi metabolites enkulu 7.5 futhi 4.5 amahora, kanye zopiclone ingashintshiwe - amahora 5.5. Cishe ama-80% of the izidakamizwa excreted nge umchamo, futhi 17-20% - ne indle.
abantu abadala izidakamizwa umzimba isibindi kancane encishisiwe. Ngaphezu kwalokho, ingxenye-ukuphila layo kungapheli angu-7. Ngokuphathelene ekuqongeleleni ketshezi asebenzayo, it is ayitholiwe at amaphilisi umthamo amaningi.
izinkomba
Okufanele ukwenze abanenkinga yokuqwasha? Odokotela batusa ukuba zibhale "Relakson". Lo mkhiqizo senzelwe ekwelapheni ezingamahlalakhona futhi eziphelayo ukuqwasha nesimo kwabadala. Futhi, ngenkuthalo esetshenziswa nalabo okunzima ngilale, Awakening ebusuku futhi ekuqaleni.
Izimo
Tablets "Relakson" is hhayi Kunconywa kulezi zimo ezilandelayo:
- hypersensitivity izidakamizwa nendaba isizinda;
- ifomu okunzima myasthenia gravis;
- ngesikhathi sokukhulelwa;
- nge elele singathatha ;
- nokuvaleka kwemigudu yokuphefumula;
- ukuhluleka ezinzima isibindi;
- ngaphansi kweminyaka eyi-18.
Izidakamizwa "Relakson": yokusetshenziswa
Ngaphambi kokuthatha amaphilisi elele Kunconywa uye kudokotela uyofuna icebiso. Kuyadingeka ukufunda imiyalelo afakiwe.
"Relakson" Tablets (igama abajwayelekile - "Zopiclone"), esithathwe ngomlomo, nje ngaphambi ukuqala ubuthongo. Abadala izidakamizwa esebenzayo yaphathwa umthamo 7.5 mg. Inani eliphelele kuyinto 15 mg ubuthongo usizo.
Ubude obuphelele ukusetshenziswa izibhebhe akufanele kube ngenyanga ezingaphezu kweyodwa. Esimweni ngasinye, isikhathi sokwelashwa kunqunywa ngamunye kuncike ngezimo zesiguli, futhi uhlobo ukuqwasha.
Phuza umuthi uma ukuqwasha ehlala kuyinto efiselekayo mayelana 3-5 izinsuku, futhi isimo - amasonto 2.5-3. Isikhathi inkambo ezingamahlalakhona ukwelashwa ukuqwasha kufanele azimisele kuphela udokotela.
Abantu abadala okungamahlala obstructive isifo samaphaphu, kanye umsebenzi kwesibindi kahle iqondiswa 3,75 mg izidakamizwa. Uma kudingeka, wathi umthamo kungase kukhule ku-7.5 mg.
Ukwelashwa nokuvikelwa ukuqwasha in iziguli esingamahlalakhona kwezinso nazo eziqala ½ i-tablet, okungukuthi, 3,75 mg.
amacala ukweqisa izidakamizwa
Ukuthatha amaphilisi amaningi okuyiluthayo kubangela CNS ukucindezeleka ntshashintshe of kobukhulu (kwi somnolence evelele esimweni ikhoma).
Ukwelashwa iqala ngokukhuphuka lavage esiswini yokweqisa. Ngokulandelayo, isiguli ezinqunyiwe sorbents.
Futhi ukwelashwa lingaze kanye nokuqapha ezibalulekile zomzimba. Izidakamizwa "Flumazenil" lisetshenziswa kuyindlela yokuvimbela.
side effects
Yiziphi imiphumela emibi is "Relakson"? Izibuyekezo ochwepheshe abanolwazi ukubika ukuthi lokhu izidakamizwa angase neqhaza ekuthuthukiseni salezi zenzakalo ezilandelayo:
- isicanucanu, ukoma futhi umunyu umlomo;
- isiyezi, ubuhlungu bekhanda, ukozela okuncane ekuseni;
- obumnandi, ulaka, ukucasuka, ukuhhema, eziya ziba zimbi kwemizwa kanye nesimo futhi bacindezeleke, kanye nokuthuthukiswa ukulahlekelwa amandla okukhumbula (kakhulu ezingavamile);
- ukulunywa, ukuqubuka, ukusabela anaphylactic (kakhulu ezingavamile);
- transaminases aphakeme isibindi futhi ane-alikhali phosphatase.
Kufanele kuphawulwe ukuthi izimo ezingavamile, izidakamizwa kubangela "khansela" syndrome, futhi ngenxa yalokho, Abuya ukuqwasha.
izidakamizwa ekuhlanganyeleni
Manje ngoba sewuyazi ukuthi yini okufanele uyenze abanenkinga yokuqwasha. Reception "Relakson" izidakamizwa kumelwe niqaphelisise, ikakhulukazi nge ukusetshenziswa ngesikhathi esisodwa neminye imithi.
Ngokusho imiyalelo, kukhuphuke umphumela inhibitory ku isimiso sezinzwa esiyinhloko zomuthi kwenzeka lihambisana antidepressant, neuroleptics, imithi ebulala izinzwa, zinhlungu, sedatives futhi hypnotics, futhi "Erythromycin" antiepileptic futhi antihistamine, analgesics kwezidakamizwa.
It is hhayi Kunconywa ukuba uphuze utshwala kanye nemithi utshwala equkethe ngesikhathi esifanayo "Relaksonom". Lokhu kungenxa yokuthi inhlanganisela enjalo ingase ithuthukise yayo umphumela okulalisayo.
Ukuthola imithi okuyiluthayo iyehlisa perfonala lokuhlushwa noma trimipramina igazi. Leli qiniso kufanele kucatshangelwe lapho isivumelwano sabo sokuhlangana kanyekanye.
izincomo Specific ukuthola okuyiluthayo
Yini odinga ukukwazi ngaphambi thatha izidakamizwa "Relakson" (efana naleli thuluzi tibalwe lapha ngentasi)?
Abantu ne ebusuku somoya ukuhlaselwa lihambisana inombolo nemithi methylxanthine amaphilisi elele kunciphisa inani ukuhlaselwa e sentathakusa, futhi kunciphisa umfutho wabo kanye nesikhathi.
Lapho ukwabela "Relakson" akufanele ngokuphelele wawususa ingozi yokulutheka. Kuye ingozi izidakamizwa kwenzeka kulezi zimo ezilandelayo:
- ayephuli imithamo kanye nesikhathi sokwelashwa;
- ngokusebenzisa kabi utshwala noma ezinye izidakamizwa;
- lapho kuhlangene utshwala noma ezinye izidakamizwa psychotropic.
Ukuze ugweme lesi sifo of "yokukhansela" ukuziyeka izidakamizwa kufanele kube elokhu enciphisa Isikali esiphansi.
Lapho ethola amaphilisi elele nesineke bangezwa ukulahlekelwa amandla okukhumbula anterograde. Ngokwejwayelekile kuzibonakalisa lapho abantu sebehlelwe ngubuthongo iphazamisekile, futhi ngemva eside isikhawu esiphakathi izidakamizwa sokuqondisa futhi sokulala.
Ukuze wehlise ezingozini ezinjalo, kubalulekile:
- Ukulala isikhathi ukunikeza okungenani amahora 6;
- ukuthatha imithi ngaphambi kokulala.
imithi Okubukwe aluboniswa ekwelapheni ukucindezeleka. Angase imaski izimpawu zaso.
umthamo ukusebenza futhi ephephile "Relaksona" ezinganeni kanye intsha engaphansi kwengu-18 ubudala engakaze zokuhlola ezasungulwa izazi. Ngakho-ke, ukuthatha izidakamizwa kulonyaka akuvunyelwe.
Uma sibheka izinkinga ezihlasela impahla kwemithi ye okuyiluthayo, kungase zibulale ikhono lesiguli ukushayela izimoto, kanye ukwenza imisebenzi enobungozi ezidinga ukunakwa anda futhi impendulo esheshayo. Kule ndaba, isikhathi sokwelashwa nale izidakamizwa kufanele siqaphelisise.
Sleeping amaphilisi "Relakson": intengo kanye analogue
Umuthi kungenziwa indawo "Relakson"? Lesi sidakamizwa, kunezindlela eziningi eziyingqayizivele. Indlela ephumelela kakhulu kukhona imithi ezilandelayo: "Milovan", "imovan", "Thorson", "Somnol", "Slipvell", "Zolinoks", "Piklodorm", ". Zopiclone"
Konke lokhu izidakamizwa, kuhlanganise "Relakson", eyakhululwa ngo-Pharmacy kuphela kadokotela. Njengoba ngentengo ke kubhekwa kusho hhayi eliphezulu kakhulu. amaphilisi 20 izidakamizwa okuyiluthayo (7.5 mg) ingatholakala for ruble 120-160.
Izibuyekezo amaphilisi elele
Ngokwe-art, izidakamizwa "Relakson" limelela kwesizukulwane sesithathu okuyiluthayo. By the way, ihlanganisa "Zaleplon" nge "zolpidem". Le mithi aphumelela kakhulu futhi ephephile ngokuphelele.
Iziguli ukubika ukuthi emva ukuphuza amaphilisi elele kakhulu baye bathuthukisa nobuthongo. Kuyilapho kulondolozwa ngokugcwele bystrofazovy sokulala wokubuyiselwa isimo ngokwengqondo nangokomzwelo.
imithi Okubukwe kunomthelela omuhle ukulala esigabeni slow wave okuyinto ebalulekile ekululameni ngokomzimba zomzimba womuntu.
Ngokwe-art, kwenza kubelula izidakamizwa esebenzayo normalizing amaphethini ubuthongo ngasiphi izinhlobo iziyaluyalu. Nokho, anakho amathuba okungenani yokuba umlutha.
Nobufakazi abonisa ukuthi iphilisi ingalali "Relakson 'ebekezelele ngokubhekakade kahle, futhi akunamthelela nezinto ezizenza nsuku zonke yomuntu. Nokho, odokotela musa batusa kokuthatha lesi umuthi. Isiguli kufanele njalo kudokotela futhi silandele yonke umthamo Kunconywa ke.
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