Impilo, Amalungiselelo
Ngempumelelo antispasmodic "Papaverine Hydrochloride"
Ukulungiselela "Papaverine hydrochloride" libhekisela miotropnym izindlela nemphumela eqinile spasmolytic. Amashumi eminyaka, isetshenziswa ukunciphisa ithoni semithambo kanye bushelelezi muscle futhi cishe zonke izitho zangaphakathi. It has a liphinyiselwe isinyathelo hypotensive. Lesi sidakamizwa dilates imithambo, kwandisa umthamo wegazi, i-cerebral ikakhulukazi. Lesi sidakamizwa ebulilini kakhulu kunciphisa excitability kwemisipha inhliziyo, kanye kunomthelela okwehlisa conductivity intracardiac. Ithonya lakhe phezu isimiso sezinzwa esiyinhloko sivezwe kancane, nakuba kunomphumela sine at ngemithamo ephakeme.
Khipha ukulungiselela "Papaverine hydrochloride" e Isikali ezifana izinhlobo:
- amaphilisi abadala 0,04g (10 nama-PC.);
- amaphilisi Wezingane of 0.01g (10 nama-PC.);
- 2% umjovo (10 ampoules);
- suppositories rectal of 20 mg (10 nama-PC.).
Izinkomba ukusetshenziswa kukhona izimo ezifana spasm ka bushelelezi imisipha izitho cholecystitis peritoneum, colic kwezinso; nesifo spastic; endarteriite; bronchospasm; pilorospazme; zibe semithambo, elise ubuchopho. Ekwelapheni angina pectoris kusho "Papaverine Hydrochloride" isetshenziselwa yokwelapha kuhlangene nezinye izidakamizwa.
Izimo ukusetshenziswa kwalesi izidakamizwa yilezi:
hypersensitivity, kahle umsebenzi sesibindi, ukufiphala kwamehlo ebuntwaneni (kufika eminyakeni engu-0.5). Asebekhulile akufanele bathathe lesi izidakamizwa ngenxa ingozi komzimba okukhulu.
Kusho "hydrochloride Papaverine": yokusetshenziswa
Umuthi wenziwa 3-4 k. ngosuku. Umthamo kwezokuphatha eyodwa amaphilisi siyahlukahluka engu-isiguli. Abadala ukhombe amaphilisi olulodwa umthamo 40-60mg. Izingane 0.5-2 g - 5mg, 3-4 PM - 5-10mg, 5-6 l. -10mg, 7-9 amalitha. - 10-15mg, 10-14 amalitha. - 15-20mg.
Umjovo iqondiswa intramuscularly noma phansi kwesikhumba. Imijovo ukwenza 2-4 k. ngelanga ngu 1-2ml. yezidakamizwa enegciwane injected kancane kakhulu ngesikhathi 20mg ngaphambilini ngokungeza nalokho sodium chloride 10-20ml (0.9% isixazululo). Le nqubo ibizwa umhlabeleli kwenziwe ngaphansi kokuqondisa kukadokotela. Ukuze oneminyaka engu-iziguli umthamo owodwa kokuqala akufanele idlule 10 mg. Ngokuvamile izidakamizwa iqondiswa parenterally lihambisana izidakamizwa ezahlukene spazmaliticheskimi kanye analgesic, ezifana izidakamizwa "Promedol".
Amakhandlela Bheka ne papaverine iqondiswa rectally, 2-3 k. 20-40mg ngosuku.
Ukulungiselela "Papaverine hydrochloride" kungase kubangele imiphumela emibi ezifana ukozela, komzimba nezinto, arrythmia ventricular, upregulation ka transaminases isibindi, wehlise blood pressure, ukuqunjelwa, eosinophilia.
Uma ukweqisa izidakamizwa waphawula izimpawu ezifana ubuthakathaka jikelele, diplopia, hypersomnia.
Ngokusebenzisa lokhu imiyalelo okukhethekile ukuze bagubhe kwezidakamizwa ukuncoma ukusetshenziswa baqaphe iziguli izidakamizwa kahle kanye nabantu abadala; abantu nge ukulimala ekhanda, i-hypothyroidism, dysfunctions adrenal, izinso kanye isibindi; tachycardia; izimo ukushaqeka.
Izidakamizwa "Papaverine hydrochloride" ngesikhathi sokukhulelwa futhi ngesikhathi ukusuthisa kungcono hhayi ukusebenzisa ngenxa ngempumelelo yalo nokuphepha lobo ayifakiwe.
Phakathi ukwelashwa, utshwala akuvunyelwe. Ukubhema ngesikhathi ukwelashwa kwehlisa ukuphumelela izidakamizwa. Bekanye ukuvuma kusho "Papaverine" futhi "Dopegitom" isinyathelo sokuqala is kakhulu ziyancipha.
Papaverine hydrochloride likhona eziningana kuhlanganiswe antispasmodics lihambisana nezinye izinto izidakamizwa:
- izidakamizwa "Lyupaverin" - ne phenobarbital;
- izidakamizwa "Pafillin" - ne platifillin gidrotata;
- ukulungiselela "Kellatrin" - ne kellinu futhi atropine sulfate ;
- izidakamizwa "Kelliverin" - ne Kellin;
- ukulungiselela "Nikoverin" - ne nicotinic acid.
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