Impilo, Amalungiselelo
"Katadolon": yokusetshenziswa, intengo, kanye nokubuyekeza. Analog "Katadolona"
Uyini izidakamizwa "Katadolon"? Analogs, intengo kanye yokusetshenziswa zomuthi izokwethulwa mathiriyeli lo sihloko. Kusukela ke uzofunda, nokuthi lokho okushiwo iyindlela, uma uneminye contraindications side effects, kulokho Lelifomu liyatholakala ekhelini equkethe e oyiyo nokunye.
Okufakiwe, ukukhululwa amafomu, ukwakheka
Izidakamizwa "Katadolon" kuqhubeka ukudayiswa amafomu ezimbili ezihlukene. incazelo yabo, ukwakheka kanye emaphaketheni, sibheka khona manje.
- Nomuthi "Katadolon Forte" - ophuzi biconvex amaphilisi okusaqanda (uhlangothi strip) equkethe ezihlukahlukene inclusions. Ukulungiswa iqukethe njengoba ingxenye esebenzayo njengoba maleate flupirtine, nezinye excipients. Tablets ezibekwe kule amabhamuza-10, 7 no-14 izingcezu, okuyinto zahlanganiswa ngo amaphakethe amakhadibhodi.
- Amaphilisi Abonayo "Katadolon kuthiye ukukhula" Unamekwe gelatin abomvu. Okuqukethwe kwezidakamizwa manje luyibhuqu lwezinyawo abe luhlaza ophuzi noma ophuzi. Omunye capsule iqukethe flupirtine maleate namanxusa ezengeziwe njengoba gelatin, magnesium stearate, amanzi, ama-titanium dioxide E172, Silicon dioxide, i-sodium lauryl sulfate, dihydrate calcium phosphate futhi copovidone. Umuthi is zahlanganiswa ngo amaphakethe amakhadibhodi 30, 50 noma 10 amaphilisi.
Isenzo kwemithi zomuthi
Ngalokho okubhekwa 'njengempi izidakamizwa futhi uma ine-analog? "Katadolon" - a analgesic-non-opioid ukuthi ine isinyathelo antispasmodic, futhi sebuningini ezahlukene analogue.
Imithi akuyona umlutha futhi uyakwazi ukunikeza umthelela eyodwa. Ngemva edonsa kuthinta G-amaprotheni, ngaleyo ndlela esishintsha umehluko okunamandla iziteshi calcium ezibangela ukuzinza the neuronal ulwelwesi ezingaba khona.
Yini izakhiwo nomuthi kubhekwe futhi okuphikisana nalo? "Katadolon" Kumele kuthathwe ngemithamo ukuthi akufanele sedlule ovumelekile esiphezulu. Kuphela kuleli cala isithako yayo asebenzayo akuphazamisi H-M-cholinergic receptor, kanye opioid, Dopamine, serotonin, futhi alfa2- receptor alpha1-adrenergic.
Ngemva kokuthola lezi amaphilisi noma amaphilisi ngaphakathi analgesia kwenzeka sibonga ukuvezwa iziteshi potassium, atholakala ezinzwa.
Ngokusho kochwepheshe, imithi nethonya elihle NMDA-receptor. Eqeda wamanje-calcium-ion, okuyinto udabula semipermeable ulwelwesi udonga.
Umgomo we isenzo izidakamizwa
Kanjani umzimba womuntu sikhuluma ngokuhoxiswa izindlela futhi okuphikisana nalo? "Katadolon" iqukethe ukubunjwa yayo flupirtine. Kuyinto yalolu ketshezi kuvimbela lasabela emsipheni ngiyibona ezintweni nociceptive. Ngenxa yalokho kuzichaya kwenzeka izinto zokubulala izinzwa.
Umuthi ayibonakali emizweni buhlungu futhi lubasize bagweme ekubeni ezingamahlalakhona. Ngaphezu kwalokho, ngempumelelo kwehlisa ubuhlungu ekhona.
Lapho eyamukelayo kusho ku muscle kwenzeka (ngenxa Ukuvinjwa izinzwa Intermediate). Asinakusho ukuthi lokhu izidakamizwa uyakwazi ukuvikela izinzwa emiphumeleni ubuthi. Ukwenza iziteshi calcium nomuthi kunciphisa okuqukethwe okulimazayo calcium ion kumaseli.
I pharmacokinetics zomuthi
Ngezinye kokuthola amaphilisi kanye amaphilisi "Katadolon kuthiye ukukhula" e emathunjini izidakamizwa izidakamizwa esebenzayo egxile ngokuphelele (90%). Ngakho-75% umthamo akheka esibindini.
Ingxenye-ukuphila umzimba kuyinto amahora 7-15. Kufika ku-70% we izidakamizwa excreted ngu izinso, kanti bonke abanye - ngokusebenzisa namathumbu.
Ngo abadala, kanye neziguli kanye kahle isibindi umsebenzi nezinso ukuqedwa isigamu-ukuphila luyanda.
Izidakamizwa "Katadolon": izinkomba ukusetshenziswa
I izinkomba ukusetshenziswa kwalesi izidakamizwa kukhona ubuhlungu Lokudabuka ehlukahlukene (okuncane noma okusesilinganisweni), okuyinto zibangelwa spasm kwemisipha bushelelezi.
Ngakho ngaphansi kwanoma iyiphi ngeziphambeko ebekiwe kubhekwa indlela futhi okuphikisana nalo? "Katadolon" livame ukusetshenziswa ubuhlungu post-op futhi ukuphathwa ikhanda, iqolo nentamo, neoplasms okubulalayo nokuhlala izimila, nokunye. D.
Izimo ukusetshenziswa kwezidakamizwa
Medicine "Katadolon" it is hhayi Kunconywa ukusebenzisa i-izinso futhi isibindi, hypoalbuminemia, umzimba wakho uxabana ne isithako esebenzayo noma izinto asizayo, tinnitus, kanye ekwelapheni asebekhulile, izingane kanye notshwala.
sokuphuzisa nomuthi
kufanele Ngithatha kanjani imithi "Katadolon"? Amaphilisi Abonayo kunoma isiphi isimo akunakwenzeka ukuhlafuna. Umthamo zomuthi ukhethwa nje umuntu ngamunye.
I zemithi elandelayo zinikwa imiyalelo exhunywe nomuthi:
- Abadala kuze iminyaka 65 enqunyiwe mg 100 zomuthi kane ngosuku (ie 1 capsule). Kufanele banamathele okufanayo zinkathi phakathi izidakamizwa imithamo. Lapho uzwakalise ubuhlungu syndrome ovunyelwe ukuthatha amaphilisi amabili kathathu ngosuku. Kumele kukhunjulwe ukuthi umthamo sangemihla kufanele kube 600 mg (okuyi 6 amaphilisi).
- Asebekhulile (engaphezu kwengu-65) izidakamizwa "Katadolon" Kufanele uthathe 100 mg kabili ngelanga. Kuye ngezinga of ubuhlungu umthamo kungenziwa lenyuke ku-300 mg ngosuku.
- Iziguli abaphethwe esingamahlalakhona kwezinso noma hypoalbuminemia, ngokuvamile iqondiswa mg ngelanga hhayi ngaphezulu kuka-300.
- Lapho nomuthi kahle umsebenzi sesibindi ayikwazi ngemithamo, okuyinto idlule 200 mg ngosuku. Isikhathi salesi ukwelashwa ingase ibe khona ehlukile. Nokho, ukwelashwa isikhathi eside kudingeka ukulawula umsebenzi enzyme isibindi.
Analogs "Katadolon" izidakamizwa aqukethe isithako ezisebenzayo ezifanayo yasekuqaleni. Nokho, lapho akhethiwe indawo, qiniseka ukuthi uxhumane nodokotela wakho bese ukhetha umthamo elikhulu.
Overdose kwezidakamizwa
Zimbalwa imibiko amacala izidakamizwa ukweqisa izidakamizwa "Katadolon" zinezinhloso ukuzibulala. Kulokhu, ubhekana zimpawu ezilandelayo: isicanucanu, esimweni prostration tachycardia, ukudideka, ukukhala, kome umlomo, ethukile.
Ekwelapheni izimpawu ezifana esetshenziswa diuresis. Ngaphezu kwalokho, isiguli unikezwe carbon ocushiwe futhi electrolyte yethulwe. Ngokweyame zonke lezi zinyathelo isimo lesiguli kuthuthukisa ngemuva kwamahora 6-12.
ukusabela ezingezinhle ngemva kokungenisa
Ezinye iziguli emva ukungenisa amaphilisi noma "Katadolon" Amaphilisi ingase ibonise ezifana side effects njengoba:
- isiyezi, ubuthakathaka, futhi ukukhathala;
- ukuqumba, isicanucanu futhi ngikhishwe ubuhlungu besisu;
- liqhaqhazela, ukuqunjelwa;
- ikhanda kanye nokukhathazeka;
- komzimba;
- izidakamizwa olubangelwa ukusha kwesibindi kohlobo;
- angaboni kahle.
Imiphumela emibi engase ivele kungalindelekile futhi kungazelelwe zinyamalale futhi phakathi ukwelashwa.
izidakamizwa ekuhlanganyeleni
Lapho kanyekanye isimiso sokuqondisa 'Katadolon "ukulungiselela kusho ezifana" Warfarin "futhi" Diazepam "isinyathelo sokuqala kungase ukugqanyiswa. Lokhu kungenxa yokuthi le mithi uxhumano nomsebenzisi kalula nge amaprotheni okukhuthaza ukufuduka lamaseli flupirtine.
Sedatives, imisipha relaxants, futhi ethanol baqinise imiphumela yabo ngaphansi kwethonya umuthi.
It is hhayi Kunconywa ukuba sihlanganise imithi nge "paracetamol", "carbamazepine" futhi "flupirtine."
Kufanele kuphawulwe ukuthi ngenkathi ukusetshenziswa kwezidakamizwa ne "coumarin" kuyadingeka ukuze ukuqapha Inkomba prothrombin.
Izixwayiso
Ngaphambi kokufaka isicelo umuthi, "Katadolon" kudingeka ufunde imiyalelo. Lithi:
- Lesi sidakamizwa kumele isetshenziswe kuphela uma abanye amaphilisi ezinhlungu yokwelapha is contraindicated.
- Phakathi isicelo se-nomuthi kubantu enciphile izinso umsebenzi kuyadingeka ukulawula lokuhlushwa creatinine egazini.
- Abantu abaneminyaka engama-65 kanye neziguli kanye hypoalbuminaemia futhi ezinzima ukungakhuli kwezinso adinga ukulungiswa umthamo izidakamizwa.
- Iziguli kufanele waxwayisa ngokuthi phakathi ukwelashwa kufanele uyinaka izimpawu isifo sesibindi. Lapho ukubonakaliswa izimpawu ezinjalo kudingeka ayeke ukuthatha izidakamizwa kanye nodokotela.
- Phakathi ukwelashwa imithi "Katadolon" kungenzeka okungamanga test asabela ngayo urobilinogen, bilirubin, ne amaprotheni ku umchamo.
- Lapho usebenzisa i-ebulilini izidakamizwa isiguli kungabonakala nasemkhakheni umchamo staining ngombala oluhlaza. Leli akulona uphawu basemtholampilo isifo.
- Phakathi ukwelashwa kubalulekile ukuba ayiyeke le imishini kanye ukushayela imoto ukulawula, kusukela iziguli zingase ziqale isiyezi futhi ukozela.
Izidakamizwa "Katadolon": analogue, ukubuyekezwa, intengo
Kuyinto efanayo nelithi ukulungiswa ithuluzi "Flugesik". Ngokuqondene esiyingqayizivele, abasolwa zihlanganisa imithi ezilandelayo: "Acupan", "Nefopam", "Milistan" futhi "Sinmeton".
Inani kubhekwe izidakamizwa kuphezulu kakhulu. Ngokuvamile, ububanzi ruble 900-1200 (kuncike ukuma kanye nenani amaphilisi, amaphilisi).
Ngokusho izimpendulo iziguli, imithi "Katadolon" ngempela ngempumelelo futhi ngokushesha ususa noma isiphi syndromes ubuhlungu. Naphezu inani elikhulu ukusabela ezingezinhle, yezidakamizwa ngokuvamile ukusebenzisa leli thuluzi ngoba ukukhululeka ubuhlungu phakathi kwemali.
Njengoba for iziguli abavamile, ezinye zazo bakhononda ngokuthi kokuthatha lesi izidakamizwa kubangela isiyezi kanye ubuthakathaka jikelele.
Ngokusho odokotela, lesi sidakamizwa "Katadolon" livame ukusetshenziswa umkhuba kuhlinzwa. Yena iyithuluzi elinamandla kakhulu, ngakho-ke akufanele kuthathwe ngaphandle udokotela.
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