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Izidakamizwa "scopolamine hydrobromide": izakhiwo, izinkomba kanye contraindications ngoba ukusetshenziswa

"Hydrobromide Scopolamine" - umuthi kabanzi lisetshenziswe imithi yesimanje. Kodwa-ke, iziguli kudingeka ulwazi olwengeziwe, ikakhulukazi izakhiwo zomuthi, izinkomba kanye contraindications ukwelashwa kanye nokunye. D.

Izidakamizwa "scopolamine hydrobromide": iresiphi, ukwakheka kanye ngesimo

Okokuqala, ake ukubhekana ekwakhiweni izidakamizwa. "Scopolamine hydrobromide" (iresiphi e-Latin - Scopolaminum Hydrobromicum) kuyinto zinhlayiya esobala kungekho nto enemibala emihle. Yiqiniso, ngokuvamile kuyabonakala ngesimo crystalline ochotshoziwe powder nge ukunambitheka okumunyu isici. Ingqikithi okubonakala kalula encibilikayo otshwaleni namanzi. By endleleni, lokhu kwakwakhe kungokwalabo iqembu alkaloids - ke lisuselwa isitshalo esifanayo njengoba atropine - a henbane, Scopoli, Belladonna, Datura.

Ekhemisi angathengwa in ifomu powder. Kodwa iningi izidakamizwa isetshenziswa ngendlela 0.05% isixazululo - bayidayise ingilazi ampoules emqulwini ka 1 ml. Kukhona izitsha eziyisikhombisa 5 noma 10 ml - isixazululo iqukethe methylcellulose Ukwakheka ezinjalo. Ampoules (noma izitsha eziyisikhombisa) kufanele agcinwe endaweni epholile, ngalolo elangeni angawi. Impilo - iminyaka 5 kusukela usuku ukwakhiwa.

Mshini wezenzo izidakamizwa

Scopolamine hydrobromide iyafana atropine mshini wezenzo - ke iyasebenza maqondana uhlelo cholinergic. Ngokwesibonelo, e isiguli ngemuva kokuthatha imithi uhlangabezana ukukhubazeka isikhashana yokuhlala, kwenhliziyo, ukwehla ngo uketshezi we nezindlala, kanye umfundi Ukuvuleka komlomo nokungcebeleka imisipha abushelelezi.

Kodwa phezu isimiso sezinzwa esiyinhloko ke izenzo ehlukile, ngenxenye ezivimbela umsebenzi wayo. Scopolamine kuvimbela ukudluliselwa nerve amaza ukuthi ngokwethemba pyramidal ipheshana motor izakhiwo emgogodleni. Ngaphezu kwalokho, amabhlogo holinoreaktivnye zemizwa kumiswa reticular. Yingakho izidakamizwa has a sine (sine) nomphumela okulalisayo kwi umzimba womuntu - encishisiwe motor umsebenzi. Phela, esinye sezici yalolu ketshezi wukuthi emva abaphathi, njengoba umthetho, kukhona ukulahlekelwa amandla okukhumbula short-term - abantu neze ukukhumbula lokho okwenzekile.

Kwezinye izimo, sebenzisa izidakamizwa? ubufakazi

I nomuthi esetshenziswa emikhakheni eminingi wezokwelapha:

  • Ngenxa sine futhi isixazululo ejenti umjovo analgesic ezisetshenziswayo ekuhlinzeni ngaphandle futhi zokubelethisa umkhuba belungiselela izinzwa.
  • Ngo Neurology inkomba ukwamukela izidakamizwa parkinsonism postencephalitic futhi shaking uhlangothi.
  • Bamehlo futhi usebenzise izidakamizwa ngesimo ngeso lehla - uma iridotsiklitah ngempumelelo futhi iritah. Amaconsi isicelo futhi uma kunesidingo ukunweba umfundi isiguli (isib ngaphambi izindlela zokuxilonga).
  • Medicine wathola isebenza wezifo zengqondo, eqinisweni izenzo njengendlela okulalisayo.
  • Nge lomoya nolwandle ukugula "scopolamine hydrobromide" kusiza ukuba sibhekane ngokuphumelelayo isicanucanu, retching bese ukwethuka. Sebenzisa le-chemical lichaza ekwakheni imithi "Aeron".

Ukusetshenziswa "scopolamine hydrobromide" kuyasiza babhekane nezinkinga eziningi. Nokho, kungaba kuphela ukhombe udokotela ukuba khona ngemva kokwenza umlando kanye kokuthola yonke idatha yokuhlola.

Izidakamizwa "scopolamine hydrobromide": yokusetshenziswa

Njengoba sekuphawuliwe, nomuthi ekhiqizwa njengoba isixazululo - iqondiswa noma phansi kwesikhumba noma intramuscularly. umthamo oqabulayo izidakamizwa (esimweni imijovo ongama) zokhahlamba kusuka 0,0002 ukuba 0,0005 g scopolamine. Ngokuvamile, iziguli iphathwa 0.5 noma 1 ml isixazululo 0.05% - imijovo banikwa izikhathi ezimbili noma ezintathu ngosuku.

Uma kuziwa iso amaconsi, iziguli iqondiswa 1-2 lehla esweni ngalinye. Inqubo kufanele liphindwe izikhathi 1-2 ngosuku, isebenzisa isisombululo 0.25%. Kuyaqondakala ukuthi umuthi anamandla futhi autocratic, ukusetshenziswa yakhe nokuwubuwula kungaholela ezinkingeni esiyingozi ngokwedlulele. Kuphela udokotela angakunika umuthi, kadokotela, ukunquma imithamo kanye nesikhathi sokwelashwa.

Ingabe ikhona imingcele ekutheni kanye contraindications?

Ingabe zonke izigaba abantu kungcono ukuba amise izidakamizwa "scopolamine hydrobromide"? Eqinisweni, i-izidakamizwa ezinye ukulinganiselwa. Ngeke inikezwe iziguli izifo eziphilayo yisimiso senhliziyo nemithambo yegazi.

Ukuze uhlu Izimo futhi zihlanganisa isifo sikashukela kanye glaucoma. Awukwazi ukusebenzisa izidakamizwa ekwelapheni iziguli yezifo indlala yegilo, ikakhulukazi i-hyperthyroidism. Amadoda wendlala hypertrophy isixazululo asebenzayo Ungase futhi zilimaze. Ukusetshenziswa kwasebekhulile kungenzeka, kodwa ukwenza kanjalo kufanele aqaphele kakhulu.

Imiphumela engemihle evela yokwelapha

Ngokwezibalo, lokhu izidakamizwa ibekezelelwe ezimweni eziningi kahle. Nokho, ezinye iziguli ziba nemiphumela emibi. Ngokwesibonelo, kungase kube ukuhlukumeza kuhlala lens futhi Ukuvuleka komlomo eziphikelelayo balezi zingane, esithinta nokuzwela ekukhanyeni, futhi acuity ezibukwayo.

Ezinye iziguli esekhala tachycardia, palpitations palpable. ukusabela ezingezinhle zihlanganisa isiyezi, nomlomo owomile, futhi izinkinga urinary. Ngezinye izikhathi ngokungalungile akhethiwe umthamo umuthi ivuselela - indoda iba sezinzwa ngaphezulu, okuyize, ukusangana ukuvela. Yiqiniso, ukubukeka iziyaluyalu ngenhla kufanele ubone udokotela, njengoba kungenzeka ukuthuthukisa ukuxakeka.

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