ImpiloAmalungiselelo

Izidakamizwa 'Atenolol Nycomed'

Ukuze izidakamizwa "Atenolol Nycomed" kukhona zamakhemikhali, wongwaqa amazwe nge igama "Atenolol". In ulimi bamakhemikhali pharmacologists ikhipha izidakamizwa selivela (RS) -4- (2-hydroxy -3- (isopropylamino) phenyl-acetamide. Tablets "Atenolol" zimelela oboevypuklye amaphilisi camera umbala omhlophe, baye umumo capsule. Umzimba main inikezwa notch for sekhefu ngakolunye uhlangothi, zikhona izimpawu AV55 futhi AV57.

Kokunye ithebhulethi, kuye ifomu ukukhululwa ingaqukatha amahlanu noma eziyikhulu namashumi amamiligremu angaba atenolol. Njengoba izingxenye asizayo esetshenziswa talc, gelatin, propylene glycol, ama-titanium dioxide, magnesium stearate, ipromeloza 2910 (15sP), corn isitashi, sodium lauryl sulfate, esindayo magnesium carbonate.

Medicine "Atenolol Nycomed" izenzo njengoba beta1-abakhethayo (cardioselective) adrenoceptor ivimbela i-ejenti, ulwelwesi eliletha ukuthula umsebenzi akuyona. Leli thuluzi ubonisa ukusebenza antianginal, antiarrhythmic futhi hypotensive. Umzimba womuntu ungakwazi ivimbela receptor beta-adrenergic kwenhliziyo, ekunciphiseni ukushukuma esivimba amanzi besigaba nozwela e autonomic isimiso sezinzwa futhi catecholamines, okuyinto aluka egazini. Medicine "Atenolol" nomthelela ekunciphiseni itheku automaticity, normalizes ukushaya kwenhliziyo kumile futhi ngesikhathi umsebenzi. Lokhu kuzole inqubo kanye excitation ka contractility esivimba amanzi, okwehlisa nomthelela AV-conduction. Ngo isicelo yayo kukhona ukwehla esivimba amanzi nomoya-mpilo funa. Kahle kuthinta ehlelekile ukusetshenziswa imithi "Atenolol" okuhloswe ngazo ukwehlisa wegazi. Ukuqina kwe-inciphise umfutho wegazi ophakeme kwenzeka ekupheleni kwesonto reception yesibili.

Ukulungiselela "Atenolol Nycomed" phezu temlomo reception indlela uyakwazi ugxile ipheshana yesisu umthamo 50-60% umthamo iqondiswa. Excreted ku umchamo kanye nengxenye-ukuphila amahora 6-7. Lezi zikhathi in iziguli ukungakhuli kwezinso, kuncike izinga filtration glomerular.

Izinkomba ngokuba umuthi "Atenolol Nycomed" kukhona izinhlobo nomfutho wegazi ophezulu kanye tachyarrhythmias (kuhlanganise itheku). Sebenzisa imithi njenge-ejenti yokuvimbela ukuhlaselwa angina.

Umthamo wansuku zonke zomuthi abadala ekwelapheni angina kanye nomfutho wegazi ophezulu ifinyelela 50-100 mg. amaphilisi Ukwamukelwa wenza izikhathi ezimbili ngosuku uma sicabangela iqiniso lokuthi umthamo wansuku zonke kumele singeqi 200 mg. Ukuze ahlanze phansi izidakamizwa kufanele kube nenani ezincane yamanzi.

Umuthi isetshenziswa ngokuhambisana esiqinile ne izincomo udokotela ukuba khona. Ukuzelapha akuvunyelwe. Umuthi 'Atenolol Nycomed "has nemiphumela engemihle. Isimiso senhliziyo nemithambo yegazi angaphendula ukubukeka bradycardia, AV-conduction thuthuva, ungase uzizwe emizweni of paresthesia nasemilenzeni abandayo, kwezinye izimo manifest izimpawu yinhliziyo. ipheshana yesisu iyaphendula ophambene isicanucanu izidakamizwa, ukuqunjelwa, uhudo, nomlomo owomile (ezingavamile), uhlelo endocrine - ukuthuthukiswa okungenzeka isimo hypoglycemic ezigulini abaphethwe isifo sikashukela, uhlelo urogenital - kungenzeka ukwehla potency. CNS ukusabela ezingezinhle bangase balwisane e ikhanda, isiyezi, izinkinga zokulala, ukucindezeleka, imizwa yokukhathala. Kungenzeka futhi ukusabela kabi komzimba, ukulunywa, futhi ububomvu. Cases okhulisa ukujuluka, ukuncishiswa izinyembezi uketshezi uketshezi zalotshwa, okuvela conjunctivitis.

Futhi, kukhona eziningi Izimo. Ohlwini yabo ihlanganisa izigaba ngazinye ezingamahlalakhona inhliziyo ukwehluleka, bradycardia, hypotension, ukuzwela kwabaningi izidakamizwa, kanye nabanye.

Gcina imithi endaweni eyomile, bavikeleke ukukhanya, ukukhishwa kwezingane. lokushisa Igumbi 25 ° C. Umuthi igcina impahla yayo iminyaka emihlanu.

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